Two etomidate sites in α1β2γ2 γ-aminobutyric acid type A receptors contribute equally and noncooperatively to modulation of channel gating.
about
Mutations at beta N265 in γ-aminobutyric acid type A receptors alter both binding affinity and efficacy of potent anestheticsCorrection for Inhibition Leads to an Allosteric Co-Agonist Model for Pentobarbital Modulation and Activation of α1β3γ2L GABAA ReceptorsPositive and Negative Allosteric Modulation of an α1β3γ2 γ-Aminobutyric Acid Type A (GABAA) Receptor by Binding to a Site in the Transmembrane Domain at the γ+-β- Interface.γ-Aminobutyric Acid Type A Receptor Modulation by Etomidate Analogs.State-dependent etomidate occupancy of its allosteric agonist sites measured in a cysteine-substituted GABAA receptor.Novel positive allosteric modulators of GABAA receptors with anesthetic activity.Cysteine substitutions define etomidate binding and gating linkages in the α-M1 domain of γ-aminobutyric acid type A (GABAA) receptorsEtomidate produces similar allosteric modulation in α1β3δ and α1β3γ2L GABA(A) receptors.Comparison of αβδ and αβγ GABAA receptors: Allosteric modulation and identification of subunit arrangement by site-selective general anesthetics.Competitive Antagonism of Anesthetic Action at the γ-Aminobutyric Acid Type A Receptor by a Novel Etomidate Analog with Low Intrinsic Efficacy.
P2860
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P2860
Two etomidate sites in α1β2γ2 γ-aminobutyric acid type A receptors contribute equally and noncooperatively to modulation of channel gating.
description
2012 nî lūn-bûn
@nan
2012年の論文
@ja
2012年論文
@yue
2012年論文
@zh-hant
2012年論文
@zh-hk
2012年論文
@zh-mo
2012年論文
@zh-tw
2012年论文
@wuu
2012年论文
@zh
2012年论文
@zh-cn
name
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@ast
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@en
type
label
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@ast
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@en
prefLabel
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@ast
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@en
P2093
P2860
P1433
P1476
Two etomidate sites in α1β2γ2 ...... modulation of channel gating.
@en
P2093
Deirdre S Stewart
Grigori Guitchounts
Stuart A Forman
P2860
P304
P356
10.1097/ALN.0B013E3182567DF3
P407
P577
2012-06-01T00:00:00Z