Truncated Nucleosides as A(3) Adenosine Receptor Ligands: Combined 2-Arylethynyl and Bicyclohexane Substitutions - Wikidata - wikimedia - TriplyDB

Truncated Nucleosides as A(3) Adenosine Receptor Ligands: Combined 2-Arylethynyl and Bicyclohexane Substitutions

Truncated Nucleosides as A(3) Adenosine Receptor Ligands: Combined 2-Arylethynyl and Bicyclohexane Substitutions

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Structural probing of off-target G protein-coupled receptor activities within a series of adenosine/adenine congeners Synthesis and evaluation of N⁶-substituted apioadenosines as potential adenosine A₃ receptor modulators.Methanocarba ring as a ribose modification in ligands of G protein-coupled purine and pyrimidine receptors: synthetic approaches.Structural sweet spot for A1 adenosine receptor activation by truncated (N)-methanocarba nucleosides: receptor docking and potent anticonvulsant activity Rigid Adenine Nucleoside Derivatives as Novel Modulators of the Human Sodium Symporters for Dopamine and Norepinephrine.Structure-Activity Analysis of Biased Agonism at the Human Adenosine A3 Receptor.Rational design of sulfonated A3 adenosine receptor-selective nucleosides as pharmacological tools to study chronic neuropathic pain.Structural Probing and Molecular Modeling of the A₃ Adenosine Receptor: A Focus on Agonist Binding.A3 Adenosine Receptors as Modulators of Inflammation: From Medicinal Chemistry to Therapy.Breakthrough in GPCR Crystallography and Its Impact on Computer-Aided Drug Design.Repurposing of a Nucleoside Scaffold from Adenosine Receptor Agonists to Opioid Receptor Antagonists

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P2860

Truncated Nucleosides as A(3) Adenosine Receptor Ligands: Combined 2-Arylethynyl and Bicyclohexane Substitutions

http://www.wikidata.org/entity/Q36377951

description

2012 nî lūn-bûn

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2012年の論文

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2012年学术文章

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2012年学术文章

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2012年学术文章

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2012年学术文章

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2012年學術文章

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2012年學術文章

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2012年學術文章

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name

Truncated Nucleosides as A(3) ...... nd Bicyclohexane Substitutions

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Truncated Nucleosides as A(3) ...... nd Bicyclohexane Substitutions

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Truncated Nucleosides as A(3) ...... nd Bicyclohexane Substitutions

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ACS Medicinal Chemistry Letters

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Truncated Nucleosides as A(3) ...... nd Bicyclohexane Substitutions

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Khai Phan

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P2860

Synthesis and pharmacological characterization of [(125)I]MRS5127, a high affinity, selective agonist radioligand for the A3 adenosine receptor

The Sonogashira reaction: a booming methodology in synthetic organic chemistry.

International Union of Basic and Clinical Pharmacology. LXXXI. Nomenclature and classification of adenosine receptors--an update

Functionalized congeners of A3 adenosine receptor-selective nucleosides containing a bicyclo[3.1.0]hexane ring system.

Impact of disrupting adenosine A₃ receptors (A₃⁻/⁻ AR) on colonic motility or progression of colitis in the mouse.

Functionally biased modulation of A(3) adenosine receptor agonist efficacy and potency by imidazoquinolinamine allosteric enhancers

Colocalization and regulated physical association of presynaptic serotonin transporters with A₃ adenosine receptors.

Inhibition of experimental auto-immune uveitis by the A3 adenosine receptor agonist CF101.

Increased neutrophil adenosine a3 receptor expression is associated with hemorrhagic shock and injury severity in trauma patients.

Structure-activity relationships of truncated C2- or C8-substituted adenosine derivatives as dual acting A₂A and A₃ adenosine receptor ligands.

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596-601

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scholarly article

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10.1021/ML300107E

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7

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3

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Kenneth A. Jacobson

Silvia Paoletta

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2012-06-11T00:00:00Z

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23145215

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3491360

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