(-)-S-[3H]CGP-12177 and its use to determine the rate constants of unlabeled beta-adrenergic antagonists.
about
Reduction in beta-adrenoceptor density in cultured rat glioma C6 cells after incubation with antidepressants is dependent upon the culturing conditions used.Intestinal elimination of ofloxacin enantiomers in the rat: evidence of a carrier-mediated process.The design, synthesis and pharmacological characterization of novel β₂-adrenoceptor antagonists.Altered sympathetic nervous system signaling in the diabetic heart: emerging targets for molecular imaging.Drug-target residence time--a case for G protein-coupled receptors.Alpha 1- and beta-adrenergic receptors in brown adipose tissue of lean (Fa/?) and obese (fa/fa) Zucker rats. Effects of cold-acclimation, sucrose feeding and adrenalectomy.Quantifying the association and dissociation rates of unlabelled antagonists at the muscarinic M3 receptor.Antipsychotic agents differ in how fast they come off the dopamine D2 receptors. Implications for atypical antipsychotic action.Functional efficacy of adenosine A₂A receptor agonists is positively correlated to their receptor residence timeSlow receptor dissociation is not a key factor in the duration of action of inhaled long-acting β2-adrenoceptor agonistsDemonstration of the suitability of CGP 12177 for in vivo studies of beta-adrenoceptors.
P2860
Q34611397-654F8459-8D64-46E8-88D0-8E6C2AF8E094Q35126874-33BC23B1-33ED-4680-B2BE-7EBCC1A6D2D6Q35216471-C9B19B13-11E9-4F1A-8DC4-E606786193F0Q36337283-8DE71837-5812-490A-A7BA-48EDE98D0183Q38189272-E597F34A-B5E0-4833-A920-4D8CDD993634Q38347859-B228BD7B-4C46-46AC-9BB1-79316D576F61Q42035222-1395C9BF-EC98-4ADA-87D6-44122AD26D2DQ42140553-74564508-0682-437E-8787-18DDCBADB293Q42246408-5189FE95-73C4-486E-940F-DAB6F533F6C7Q42283741-3FF9E7AF-9D47-43A1-AF0C-B92B358DFA32Q42920670-D49A3B51-4E24-4FF4-91E9-2C4D4A38CBC2
P2860
(-)-S-[3H]CGP-12177 and its use to determine the rate constants of unlabeled beta-adrenergic antagonists.
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on February 1985
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
(-)-S-[3H]CGP-12177 and its us ...... d beta-adrenergic antagonists.
@en
type
label
(-)-S-[3H]CGP-12177 and its us ...... d beta-adrenergic antagonists.
@en
prefLabel
(-)-S-[3H]CGP-12177 and its us ...... d beta-adrenergic antagonists.
@en
P2093
P2860
P356
P1476
(-)-S-[3H]CGP-12177 and its us ...... d beta-adrenergic antagonists.
@en
P2093
P2860
P304
P356
10.1073/PNAS.82.3.925
P407
P577
1985-02-01T00:00:00Z