Small-molecule inhibitors binding to protein kinase. Part II: the novel pharmacophore approach of type II and type III inhibition.

Small-molecule inhibitors binding to protein kinase. Part II: the novel pharmacophore approach of type II and type III inhibition.

Item
http://www.wikidata.org/entity/Q38090664
Discovery of a novel mode of protein kinase inhibition characterized by the mechanism of inhibition of human mesenchymal-epithelial transition factor (c-Met) protein autophosphorylation by ARQ 197Structure-kinetic relationship study of CDK8/CycC specific compoundsIdentification of type-II inhibitors using kinase structuresSmall molecule c-Met kinase inhibitors: a review of recent patents.Development and strategies of VEGFR-2/KDR inhibitors.Targeting the DFG-in kinase conformation: a new trend emerging from a patent analysis.p38α mitogen-activated protein kinase inhibitors, a patent review (2005-2011).c-Jun N-terminal kinase inhibitors: a patent review (2010 - 2014).Rational design, synthesis, and biological evaluation of Pan-Raf inhibitors to overcome resistance.Bisarylureas Based on 1H-Pyrazolo[3,4-d]pyrimidine Scaffold as Novel Pan-RAF Inhibitors with Potent Anti-Proliferative Activities: Structure-Based Design, Synthesis, Biological Evaluation and Molecular Modelling Studies.Synthesis and p38 Inhibitory Activity of Some Novel Substituted N,N'-Diarylurea Derivatives.Ribosomal S6 kinase (RSK) modulators: a patent review.Inferring multi-target QSAR models with taxonomy-based multi-task learning.A Comprehensive Structural Overview of p38α Mitogen-Activated Protein Kinase in Complex with ATP-Site and Non-ATP-Site Binders.A multistep docking and scoring protocol for congeneric series: Implementation on kinase DFG-out type II inhibitors.Application of shape-based and pharmacophore-based in silico screens for identification of Type II protein kinase inhibitors.
P2860

Small-molecule inhibitors binding to protein kinase. Part II: the novel pharmacophore approach of type II and type III inhibition.

Item
http://www.wikidata.org/entity/Q38090664
description
article científic
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article scientifique
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articol științific
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articolo scientifico
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artigo científico
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artigo científico
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artigo científico
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artikel ilmiah
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artículo científico
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Small-molecule inhibitors bind ...... pe II and type III inhibition.
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type
label
Small-molecule inhibitors bind ...... pe II and type III inhibition.
@en
prefLabel
Small-molecule inhibitors bind ...... pe II and type III inhibition.
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P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P698
P356
P1433
P1476
Small-molecule inhibitors bind ...... pe II and type III inhibition.
@en
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P698