Synthesis, biological evaluation, and computational studies of Tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.
about
Multiple Targeting Approaches on Histamine H3 Receptor AntagonistsRecent development of multifunctional agents as potential drug candidates for the treatment of Alzheimer's disease.Procognitive properties of drugs with single and multitargeting H3 receptor antagonist activities.Rational Modification of the Biological Profile of GPCR Ligands through Combination with Other Biologically Active Moieties.Molecular Modelling Approaches for the Analysis of Histamine Receptors and Their Interaction with Ligands.Mathematical analysis of the sodium sensitivity of the human histamine H3 receptorAminobenzimidazoles and Structural Isomers as Templates for Dual-Acting Butyrylcholinesterase Inhibitors and hCB2 R Ligands To Combat Neurodegenerative Disorders.Biatractylolide Modulates PI3K-Akt-GSK3β-Dependent Pathways to Protect against Glutamate-Induced Cell Damage in PC12 and SH-SY5Y Cells.Progress in the development of histamine H3 receptor antagonists/inverse agonists: a patent review (2013-2017).Investigation of naphthofuran moiety as potential dual inhibitor against BACE-1 and GSK-3β: molecular dynamics simulations, binding energy, and network analysis to identify first-in-class dual inhibitors against Alzheimer's disease.Synthesis and Biological Assessment of Racemic Benzochromenopyrimidinimines as Antioxidant, Cholinesterase, and Aβ1-42 Aggregation Inhibitors for Alzheimer's Disease Therapy.
P2860
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P2860
Synthesis, biological evaluation, and computational studies of Tri- and tetracyclic nitrogen-bridgehead compounds as potent dual-acting AChE inhibitors and hH3 receptor antagonists.
description
2014 nî lūn-bûn
@nan
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
2014年论文
@zh
2014年论文
@zh-cn
name
Synthesis, biological evaluati ...... and hH3 receptor antagonists.
@en
type
label
Synthesis, biological evaluati ...... and hH3 receptor antagonists.
@en
prefLabel
Synthesis, biological evaluati ...... and hH3 receptor antagonists.
@en
P2093
P2860
P356
P1476
Synthesis, biological evaluati ...... s and hH3 receptor antagonists
@en
P2093
Andrea Strasser
Christoph A Sotriffer
Fouad H Darras
Hans-Joachim Wittmann
Martin Nimczick
Michael Decker
Sarah Wehle
Steffen Pockes
P2860
P304
P356
10.1021/CN4002126
P577
2014-01-14T00:00:00Z