Identification of New Nonsteroidal RORα Ligands; Related Structure-Activity Relationships and Docking Studies.

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Discovery and structural optimization of 4-(4-(benzyloxy)phenyl)-3,4-dihydropyrimidin-2(1H)-ones as RORc inverse agonists.

P2860

Q37399370-D3D66E79-3333-44F7-A302-D982B088D49A

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Identification of New Nonsteroidal RORα Ligands; Related Structure-Activity Relationships and Docking Studies.

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http://www.wikidata.org/entity/Q39778851

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2013 nî lūn-bûn

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2013年の論文

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2013年学术文章

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2013年学术文章

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2013年学术文章

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Identification of New Nonstero ...... tionships and Docking Studies.

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Identification of New Nonstero ...... tionships and Docking Studies.

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type

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label

Identification of New Nonstero ...... tionships and Docking Studies.

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Identification of New Nonstero ...... tionships and Docking Studies.

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Identification of New Nonstero ...... tionships and Docking Studies.

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Identification of New Nonstero ...... tionships and Docking Studies.

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P1476

Identification of New Nonstero ...... ationships and Docking Studies

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P2093

Christophe Berini

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Jean-François Delhomel

http://www.w3.org/2001/XMLSchema#string

Lionel Colliandre

http://www.w3.org/2001/XMLSchema#string

Luc Morin-Allory

http://www.w3.org/2001/XMLSchema#string

Lucie Maingot

http://www.w3.org/2001/XMLSchema#string

Mathieu Dubernet

http://www.w3.org/2001/XMLSchema#string

Matthieu Daillet

http://www.w3.org/2001/XMLSchema#string

Robert Walczak

http://www.w3.org/2001/XMLSchema#string

Stéphane Helleboid

http://www.w3.org/2001/XMLSchema#string

Sylvain Routier

http://www.w3.org/2001/XMLSchema#string

P2860

Modulation of retinoic acid receptor-related orphan receptor alpha and gamma activity by 7-oxygenated sterol ligands

X-ray structure of the hRORalpha LBD at 1.63 A: structural and functional data that cholesterol or a cholesterol derivative is the natural ligand of RORalpha

Crystal structure of the human RORalpha Ligand binding domain in complex with cholesterol sulfate at 2.2 A

Glide: a new approach for rapid, accurate docking and scoring. 1. Method and assessment of docking accuracy

Absence of the SRC-2 coactivator results in a glycogenopathy resembling Von Gierke's disease

A second class of nuclear receptors for oxysterols: Regulation of RORalpha and RORgamma activity by 24S-hydroxycholesterol (cerebrosterol)

Staggerer, a new mutation in the mouse affecting the cerebellum.

Disruption of the nuclear hormone receptor RORalpha in staggerer mice.

Identification of SR1078, a synthetic agonist for the orphan nuclear receptors RORα and RORγ.

Identification of SR3335 (ML-176): a synthetic RORα selective inverse agonist

P304

504-508

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scholarly article

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10.1021/ML300471D

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P478

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Nicolas Duguet

Marilyne Bourotte

P577

2013-04-10T00:00:00Z

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24900700

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P932

4027490

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Identification of New Nonsteroidal RORα Ligands; Related Structure-Activity Relationships and Docking Studies.

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P2860

P2860

Identification of New Nonsteroidal RORα Ligands; Related Structure-Activity Relationships and Docking Studies.

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P1433

P1476

P2093

P2860

P304

P31

P356

P433

P478

P50

P577

P698

P932

P356

P1433

P1476

P2093

P2860

P304

P31

P356

P433

P478

P50

P577

P698

P932