Inhibition of rabbit brain prolyl endopeptidase by n-benzyloxycarbonyl-prolyl-prolinal, a transition state aldehyde inhibitor.
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Multiple myelomaThe Dipeptidyl Peptidase Family, Prolyl Oligopeptidase, and Prolyl Carboxypeptidase in the Immune System and Inflammatory Disease, Including AtherosclerosisStructural analysis of prolyl oligopeptidases using molecular docking and dynamics: insights into conformational changes and ligand bindingAcute kidney injury in the rat causes cardiac remodelling and increases angiotensin-converting enzyme 2 expressionRelease of vasopressin from the rat hypothalamo-neurohypophysial system by angiotensin-(1-7) heptapeptide.Targeting prolyl endopeptidase with valproic acid as a potential modulator of neutrophilic inflammationNeurotensin increases mortality and mast cells reduce neurotensin levels in a mouse model of sepsis.Mass spectrometry for the molecular imaging of angiotensin metabolism in kidney.Comparative analysis of the substrate preferences of two post-proline cleaving endopeptidases, prolyl oligopeptidase and fibroblast activation protein α.Intracellular activation and deactivation of tasidotin, an analog of dolastatin 15: correlation with cytotoxicityProlylcarboxypeptidase regulates food intake by inactivating alpha-MSH in rodents.Degradation of thyrotropin-releasing hormone and luteinising hormone-releasing hormone by enzymes of brain tissue.Low molecular weight inhibitors of Prolyl Oligopeptidase: a review of compounds patented from 2003 to 2010.Prolyl oligopeptidase and its role in the organism: attention to the most promising and clinically relevant inhibitors.Mycobacterium tuberculosis Prolyl Oligopeptidase Induces In vitro Secretion of Proinflammatory Cytokines by Peritoneal Macrophages.Herbimycin A induces the 20 S proteasome- and ubiquitin-dependent degradation of receptor tyrosine kinases.Slow tight-binding inhibition of prolyl endopeptidase by benzyloxycarbonyl-prolyl-prolinal.Benzyloxycarbonylprolylprolinal, a transition-state analogue for prolyl oligopeptidase, forms a tetrahedral adduct with catalytic serine, not a reactive cysteine.Prolyl oligopeptidase is involved in release of the antifibrotic peptide Ac-SDKP.High-affinity receptor sites and rapid proteolytic inactivation of neurotensin in primary cultured neurons.Neurotensin-metabolizing peptidases in rat fundus plasma membranes.Activation of phosphatidylinositol turnover by neurotensin receptors in the human colonic adenocarcinoma cell line HT29.Novel proline endopeptidase inhibitors do not modify Abeta40/42 formation and degradation by human cells expressing wild-type and swedish mutated beta-amyloid precursor protein.Specificity of prolyl endopeptidase.Synthesis and inhibitory activity of acyl-peptidyl-pyrrolidine derivatives toward post-proline cleaving enzyme; a study of subsite specificity.Murine T cells expressing high activity of prolyl endopeptidase are susceptible to activation-induced cell death.Synthesis and inhibitory activity of acyl-peptidyl-prolinalderivatives toward post-proline cleaving enzyme as nootropic agents.
P2860
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P2860
Inhibition of rabbit brain prolyl endopeptidase by n-benzyloxycarbonyl-prolyl-prolinal, a transition state aldehyde inhibitor.
description
1983 nî lūn-bûn
@nan
1983年の論文
@ja
1983年論文
@yue
1983年論文
@zh-hant
1983年論文
@zh-hk
1983年論文
@zh-mo
1983年論文
@zh-tw
1983年论文
@wuu
1983年论文
@zh
1983年论文
@zh-cn
name
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@en
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@nl
type
label
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@en
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@nl
prefLabel
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@en
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@nl
P2860
P1476
Inhibition of rabbit brain pro ...... tion state aldehyde inhibitor.
@en
P2093
P2860
P356
10.1111/J.1471-4159.1983.TB11815.X
P407
P577
1983-07-01T00:00:00Z