Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
about
A new experimental model for assessing drug efficacy against Trypanosoma cruzi infection based on highly sensitive in vivo imagingNon-invasive in vivo study of the Trypanosoma vivax infectious process consolidates the brain commitment in late infectionsHuprines as a new family of dual acting trypanocidal-antiplasmodial agentsMethodological advances in drug discovery for Chagas disease.Megazol and its bioisostere 4H-1,2,4-triazole: comparing the trypanocidal, cytotoxic and genotoxic activities and their in vitro and in silico interactions with the Trypanosoma brucei nitroreductase enzyme.Bioluminescence imaging of chronic Trypanosoma cruzi infections reveals tissue-specific parasite dynamics and heart disease in the absence of locally persistent infection.Targeting the substrate preference of a type I nitroreductase to develop antitrypanosomal quinone-based prodrugs.Evaluating 5-nitrofurans as trypanocidal agents.Evaluating aziridinyl nitrobenzamide compounds as leishmanicidal prodrugsSynthesis and biological evaluation of N-cyanoalkyl-, N-aminoalkyl-, and N-guanidinoalkyl-substituted 4-aminoquinoline derivatives as potent, selective, brain permeable antitrypanosomal agents.Multicomponent reaction-based synthesis and biological evaluation of tricyclic heterofused quinolines with multi-trypanosomatid activityLuminescent multiplex viability assay for Trypanosoma brucei gambiense.Novel 3-nitro-1H-1,2,4-triazole-based compounds as potential anti-Chagasic drugs: in vivo studiesTransformation of saturated nitrogen-containing heterocyclic compounds by microorganisms.Novel drug discovery for Chagas disease.Further insights into biological evaluation of new anti-Trypanosoma cruzi 5-nitroindazoles.Novel 3-nitro-1H-1,2,4-triazole-based piperazines and 2-amino-1,3-benzothiazoles as antichagasic agentsNovel 3-nitro-1H-1,2,4-triazole-based amides and sulfonamides as potential antitrypanosomal agents.A class of 5-nitro-2-furancarboxylamides with potent trypanocidal activity against Trypanosoma brucei in vitro.Nifurtimox activation by trypanosomal type I nitroreductases generates cytotoxic nitrile metabolites.Novel 3-nitro-1H-1,2,4-triazole-based aliphatic and aromatic amines as anti-chagasic agents.Pharmacokinetics of hydroxymethylnitrofurazone, a promising new prodrug for Chagas' disease treatmentAldo-keto reductase and alcohol dehydrogenase contribute to benznidazole natural resistance in Trypanosoma cruzi.Tetrasubstituted Imidazolium Salts as Potent Antiparasitic Agents against African and American Trypanosomiases.Unravelling the role of SNM1 in the DNA repair system of Trypanosoma brucei.
P2860
Q27011506-D7313C02-80CA-4A0E-BA0E-9774B008C0B6Q28484843-EF73A95D-D243-436A-80BE-7F00D4C353B5Q33818962-0D4950F4-9702-4E94-A0CB-BA169886BDD6Q33945347-E9B87003-D67E-499C-B3D4-489E57B423F5Q34040586-4486E067-DC2B-4645-B51C-1B99C0464143Q34310471-473877B6-CCD5-4A38-821A-12DDF682C4DCQ34403287-1B43CB09-3156-4D9E-AF5A-5C23834A7619Q34555495-C841961E-110C-41C1-8008-D7250906B844Q35027309-BDD08877-17F3-4049-8AF0-2E74A5D2E7B8Q36122310-D9B6FC20-3730-48F3-A3BC-84155F236D23Q36263511-ED0E8E52-4016-4302-B88A-84A6CEE03E3BQ37057168-9B94B7BE-C8A6-4C67-A029-51D01CE46402Q37628155-12FE111C-74F4-4BB5-AC92-A78F01A55297Q38172427-E9EE728D-1AA3-407A-8DC4-00A2252D8A7BQ38770142-B9D64BE4-238A-48C8-A088-B44D1D0204F6Q39033607-4282BA15-9DA5-446B-BD3E-1C1A1F0B55B3Q39099136-CCE6E52F-2496-4C29-9580-DA1958734EEFQ39355235-9A3BE78C-992E-479D-A21E-EBD6CF1FFF02Q39492522-08B92B94-9B66-41F8-8814-24E339797BE7Q39587113-4F1EBA2E-53B2-4A9E-96AF-99FA2B6311CEQ40394480-7EC88A18-9D7A-4B26-9D3D-948D0A518133Q42098034-71DA99C2-D080-4A45-B933-5A7DCE828627Q46310403-2BC7CF6C-E6F7-489E-8DDB-171C04E5077FQ48235808-E1ECB35B-DEE3-4E21-AB65-FE039B2E72B7Q52657468-C2440E5C-BE48-428C-8652-698C8B94E743
P2860
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
description
2010 nî lūn-bûn
@nan
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
2010年论文
@zh
2010年论文
@zh-cn
name
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@en
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@nl
type
label
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@en
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@nl
prefLabel
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@en
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@nl
P2093
P2860
P50
P921
P356
P1476
Trypanocidal activity of aziridinyl nitrobenzamide prodrugs.
@en
P2093
Noosheen Bashir
Shane R Wilkinson
P2860
P304
P356
10.1128/AAC.00800-10
P407
P577
2010-08-02T00:00:00Z