Synthesis and biological evaluation of the first pentafluorosulfanyl analogs of mefloquine.
about
A small-fish model for behavioral-toxicological screening of new antimalarial drugs: a comparison between erythro- and threo-mefloquine.Pentafluorosulfanyl-containing flufenamic acid analogs: Syntheses, properties and biological activitiesStructure-Activity Study of Bioisosteric Trifluoromethyl and Pentafluorosulfanyl Indole Inhibitors of the AAA ATPase p97.Recent advances in fluorination techniques and their anticipated impact on drug metabolism and toxicity.Application of the Pentafluorosulfanyl Group as a Bioisosteric Replacement.Synthesis and evaluation of 7-substituted 4-aminoquinoline analogues for antimalarial activity.Synthesis of SF5-containing benzisoxazoles, quinolines, and quinazolines by the Davis reaction of nitro-(pentafluorosulfanyl)benzenes.Evaluation of tert-butyl isosteres: case studies of physicochemical and pharmacokinetic properties, efficacies, and activities.Synthesis of Phthalocyanines with a Pentafluorosulfanyl Substituent at Peripheral Positions.Optimized quinoline amino alcohols as disruptors and dispersal agents of Vibrio cholerae biofilms.Synthesis and reactivity of aliphatic sulfur pentafluorides from substituted (pentafluorosulfanyl)benzenes.Microbial biotransformation of aryl sulfanylpentafluorides.Trapped in misbelief for almost 40 years: selective synthesis of the four stereoisomers of mefloquine.SF5-Pyridylaryl-λ3-iodonium salts and their utility as electrophilic reagents to access SF5-pyridine derivatives in the late-stage of synthesis.Formation of α-SF5-Enolate Enables Preparation of 3-SF5-Quinolin-2-ones, 3-SF5-Quinolines, and 3-SF5-Pyridin-2-ones: Evaluation of their Physicochemical Properties.Silver-induced self-immolative Cl-F exchange fluorination of arylsulfur chlorotetrafluorides: synthesis of arylsulfur pentafluorides.Allosteric agonists of the calcium receptor (CaR): fluorine and SF5 analogues of cinacalcet.Synthesis and Evaluation of Potent KCNQ2/3-Specific Channel Activators.Simultaneous introduction of trifluoromethyl and λ(6)-pentafluorosulfanyl substituents using F5S-C≡C-CF3 as a dienophile.Racemic and enantioselective metal-catalyzed synthesis of SF5-containing diarylmethanols.Preparations of SF(5)- and CF(3)-substituted arenes utilizing the 7-oxabicyclo[2.2.1]hept-2-ene synthones.
P2860
Q35606501-B23030DC-FD59-4309-9708-CA0EF6126AE7Q36142192-CDCD6ECA-AD30-4928-A5CB-B3413C49A5C7Q36367307-23C5857B-86B8-46E2-8412-5265F206834FQ38366495-DC83B9C9-8858-4B96-B6F7-F129A95A4034Q38637720-E6DA231F-8E82-4683-B1A7-418990A3E528Q39475539-DB03A796-E575-4B6C-8D71-353256D8CF07Q41190221-E81F1208-2850-4CC0-BE02-EB5BDC8981B3Q41512872-719E9A22-510B-4562-9B67-3874ACD95A45Q41791511-D19EBBF0-2014-4F18-BEB0-80287DF309F2Q41887959-939BA97E-0191-4BAB-9840-B6AB9EA2955FQ42237305-69CAFB0F-8922-49AC-ABDC-C1308B352CD5Q43689368-ECE0A9B8-5894-479F-AEE1-F0FC7149EADDQ44083782-C84E8E81-4C52-424C-8119-C4882E54C7A3Q48106643-5904B390-EE93-4DA0-A6FB-EF1E6E7C29DFQ48269510-ED4453BE-5B6C-459D-B4C2-0AF06A81A084Q48629344-2B5E4D62-ED6F-48C2-9D7C-0BF8F73D44F5Q50058484-C0DBF206-3E16-4071-92CD-8AED3C7DF62FQ51738570-59190922-147B-4FC3-B8C7-A470B028B4AEQ52867389-05D16373-EF28-4674-BFFE-F133028D1FBCQ54342459-5A70280E-05D5-47B6-A611-50E47589CBBEQ54678491-2650CF88-CD3C-483A-A062-716CC2902DE2
P2860
Synthesis and biological evaluation of the first pentafluorosulfanyl analogs of mefloquine.
description
2009 nî lūn-bûn
@nan
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
2009年论文
@zh
2009年论文
@zh-cn
name
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@en
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@nl
type
label
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@en
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@nl
prefLabel
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@en
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@nl
P2093
P2860
P356
P1476
Synthesis and biological evalu ...... ulfanyl analogs of mefloquine.
@en
P2093
Diana Caridha
Erin E Milner
Geoffrey S Dow
Lucia Gerena
Norma Roncal
Steven J Geib
Tingting Mo
P2860
P304
P356
10.1039/B911483A
P50
P577
2009-08-07T00:00:00Z