IC50-based approaches as an alternative method for assessment of time-dependent inhibition of CYP3A4.
about
ICECAP: an integrated, general-purpose, automation-assisted IC50/EC50 assay platform.p53: key conductor of all anti-acne therapies.Exploring the Role of CYP3A4 Mediated Drug Metabolism in the Pharmacological Modulation of Nitric Oxide Production.Drug-drug interaction potential of marketed oncology drugs: in vitro assessment of time-dependent cytochrome P450 inhibition, reactive metabolite formation and drug-drug interaction prediction.Single concentration loss of activity assay provides an improved assessment of drug-drug interaction risk compared to IC50-shift.
P2860
IC50-based approaches as an alternative method for assessment of time-dependent inhibition of CYP3A4.
description
2010 nî lūn-bûn
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2010年の論文
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年学术文章
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2010年學術文章
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name
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
@en
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
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type
label
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
@en
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
@nl
prefLabel
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
@en
IC50-based approaches as an al ...... ependent inhibition of CYP3A4.
@nl
P2860
P1433
P1476
IC50-based approaches as an al ...... dependent inhibition of CYP3A4
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P2093
Howard J Burt
J Brian Houston
P2860
P304
P356
10.3109/00498251003698555
P407
P577
2010-05-01T00:00:00Z