Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.
about
Generation and screening of oxime libraries addressing the neuronal GABA transporter GAT1.Astrocytic Control of Biosynthesis and Turnover of the Neurotransmitters Glutamate and GABA.The GABA synapse as a target for antiepileptic drugs: a historical overview focused on GABA transporters.A binding mode hypothesis of tiagabine confirms liothyronine effect on γ-aminobutyric acid transporter 1 (GAT1)Conformationally Restricted GABA with Bicyclo[3.1.0]hexane Backbone as the First Highly Selective BGT-1 Inhibitor.Astrocytic GABA Transporters: Pharmacological Properties and Targets for Antiepileptic Drugs.Glial GABA Transporters as Modulators of Inhibitory Signalling in Epilepsy and Stroke.Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements.Pharmacological identification of a guanidine-containing β-alanine analogue with low micromolar potency and selectivity for the betaine/GABA transporter 1 (BGT1).
P2860
Q35393157-31E0DC4A-C6B5-4D12-A9D3-A7994D14707BQ38130674-01B9C50F-657A-4FB8-B3F7-B0F330CF8510Q38195817-0E368400-DBA1-4865-A92E-C1389E0CA8C7Q41439937-D1C59352-6BDA-4F5F-8175-5B402791EC61Q41817527-2AEC0284-89A5-4A23-9A62-838B3351634BQ46318123-A700519D-0CE8-48B0-9F3E-153AA3AF9D23Q47923163-18942708-5973-4422-BEF5-4222C866B1A9Q48144959-CAAF9726-A555-4E3D-BD75-6AE0A3E8E815Q48774964-433D4698-1483-46F6-9806-0524E6E2903A
P2860
Selective mGAT2 (BGT-1) GABA uptake inhibitors: design, synthesis, and pharmacological characterization.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年学术文章
@wuu
2013年学术文章
@zh
2013年学术文章
@zh-cn
2013年学术文章
@zh-hans
2013年学术文章
@zh-my
2013年学术文章
@zh-sg
2013年學術文章
@yue
2013年學術文章
@zh-hant
name
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@en
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@nl
type
label
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@en
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@nl
prefLabel
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@en
Selective mGAT2 (BGT-1) GABA u ...... rmacological characterization.
@nl
P2093
P50
P356
P1476
Selective mGAT2 (BGT-1) GABA u ...... armacological characterization
@en
P2093
H Steve White
Jonas Skovgaard-Petersen
Karsten K Madsen
Lars Jørgensen
Nrupa Borkar
Povl Krogsgaard-Larsen
Stine B Vogensen
P304
P356
10.1021/JM301872X
P407
P577
2013-02-27T00:00:00Z