Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues.
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Drug and cell type-specific regulation of genes with different classes of estrogen receptor beta-selective agonistsEstrogen receptor beta-selective agonists stimulate calcium oscillations in human and mouse embryonic stem cell-derived neuronsRegulation of specific target genes and biological responses by estrogen receptor subtype agonistsThe hop phytoestrogen, 8-prenylnaringenin, reverses the ovariectomy-induced rise in skin temperature in an animal model of menopausal hot flushesDifferential neuroprotective and antiinflammatory effects of estrogen receptor (ER)alpha and ERbeta ligand treatmentWhat's new in estrogen receptor action in the female reproductive tractSex steroid hormones matter for learning and memory: estrogenic regulation of hippocampal function in male and female rodentsPancreatic insulin content regulation by the estrogen receptor ER alphaCyclopia extracts act as ERα antagonists and ERβ agonists, in vitro and in vivoEstrogen replacement therapy-induced neuroprotection against brain ischemia-reperfusion injury involves the activation of astrocytes via estrogen receptor β.Estrogen Receptor β in Melanoma: From Molecular Insights to Potential Clinical UtilityDifferential ligand binding affinities of human estrogen receptor-α isoformsEstrogen-induced smooth muscle cell growth is regulated by tuberin and associated with altered activation of platelet-derived growth factor receptor-beta and ERK-1/2Estrogen receptor alpha and beta specific agonists regulate expression of synaptic proteins in rat hippocampusThe roles of membrane estrogen receptor subtypes in modulating dopamine transporters in PC-12 cellsEstrogen modulates TNF-alpha-induced inflammatory responses in rat aortic smooth muscle cells through estrogen receptor-beta activationAn ADIOL-ERβ-CtBP transrepression pathway negatively regulates microglia-mediated inflammationEstrogenic plant extracts reverse weight gain and fat accumulation without causing mammary gland or uterine proliferationFatty acids derived from royal jelly are modulators of estrogen receptor functionsEstrogen receptor-β regulates human tryptophan hydroxylase-2 through an estrogen response element in the 5' untranslated regionNudging oligodendrocyte intrinsic signaling to remyelinate and repair: Estrogen receptor ligand effects.Estrogen receptor β ligand therapy activates PI3K/Akt/mTOR signaling in oligodendrocytes and promotes remyelination in a mouse model of multiple sclerosis.Chronic treatment with estrogen receptor agonists restores acquisition of a spatial learning task in young ovariectomized rats.Estrogen receptor-beta agonist diarylpropionitrile: biological activities of R- and S-enantiomers on behavior and hormonal response to stress.Resting intracellular calcium concentration, depolarizing Gamma-Aminobutyric Acid and possible role of local estradiol synthesis in the developing male and female hippocampusThe immunophilin-like protein XAP2 is a negative regulator of estrogen signaling through interaction with estrogen receptor αNeuroprotective and anti-inflammatory effects of estrogen receptor ligand treatment in mice.The Concise Guide to PHARMACOLOGY 2013/14: nuclear hormone receptors.Identification of ligands with bicyclic scaffolds provides insights into mechanisms of estrogen receptor subtype selectivity.Extra-nuclear signalling of estrogen receptor to breast cancer cytoskeletal remodelling, migration and invasionBiphenyl C-cyclopropylalkylamides: New scaffolds for targeting estrogen receptor betaNew stably transfected bioluminescent cells expressing FLAG epitope-tagged estrogen receptors to study their chromatin recruitment.Estrogen receptor hormone agonists limit trauma hemorrhage shock-induced gut and lung injury in rats.Activation of a Gq-coupled membrane estrogen receptor rapidly attenuates α2-adrenoceptor-induced antinociception via an ERK I/II-dependent, non-genomic mechanism in the female ratESR1 and ESR2 differentially regulate daily and circadian activity rhythms in female mice.Regulation of aryl hydrocarbon receptor function by selective estrogen receptor modulators.An additive interaction between the NFkappaB and estrogen receptor signalling pathways in human endometrial epithelial cells.Activation of estrogen receptor α enhances bradykinin signaling in peripheral sensory neurons of female ratsEstrogen: a master regulator of bioenergetic systems in the brain and bodyMinireview: Estrogen receptor-beta: mechanistic insights from recent studies.
P2860
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P2860
Estrogen receptor-beta potency-selective ligands: structure-activity relationship studies of diarylpropionitriles and their acetylene and polar analogues.
description
2001 nî lūn-bûn
@nan
2001年の論文
@ja
2001年学术文章
@wuu
2001年学术文章
@zh
2001年学术文章
@zh-cn
2001年学术文章
@zh-hans
2001年学术文章
@zh-my
2001年学术文章
@zh-sg
2001年學術文章
@yue
2001年學術文章
@zh-hant
name
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@en
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@nl
type
label
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@en
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@nl
prefLabel
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@en
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@nl
P2093
P356
P1476
Estrogen receptor-beta potency ...... acetylene and polar analogues.
@en
P2093
Carlson KE
Katzenellenbogen BS
Katzenellenbogen JA
Marriner GA
P304
P356
10.1021/JM010254A
P407
P577
2001-11-01T00:00:00Z