High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 receptors.
about
Modeling ligand recognition at the P2Y12 receptor in light of X-ray structural information.The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsPharmacochemistry of the platelet purinergic receptors.Ticlopidine in its prodrug form is a selective inhibitor of human NTPDase1Central P2Y12 receptor blockade alleviates inflammatory and neuropathic pain and cytokine production in rodents.Comparison of three GPCR structural templates for modeling of the P2Y12 nucleotide receptor.Targeting renal purinergic signalling for the treatment of lithium-induced nephrogenic diabetes insipidus.Morphological and Molecular Characterization of Human Dermal Lymphatic CollectorsP2Y12 Receptor Localizes in the Renal Collecting Duct and Its Blockade Augments Arginine Vasopressin Action and Alleviates Nephrogenic Diabetes Insipidus.Molecular Structure of P2Y Receptors: Mutagenesis, Modeling, and Chemical Probes.Recent applications of microwave irradiation to medicinal chemistry.Generation and characterization of polyclonal and monoclonal antibodies to human NTPDase2 including a blocking antibody.Anthraquinones As Pharmacological Tools and Drugs.The platelet P2Y(12) receptor under normal and pathological conditions. Assessment with the radiolabeled selective antagonist [(3)H]PSB-0413.5-alkyl-1,3-oxazole derivatives of 6-amino-nicotinic acids as alkyl ester bioisosteres are antagonists of the P2Y12 receptor.8-BuS-ATP derivatives as specific NTPDase1 inhibitors.Development of a comprehensive set of P2 receptor pharmacological research compoundsSyntheses of 2-substituted 1-amino-4-bromoanthraquinones (bromaminic acid analogues) - precursors for dyes and drugs.Competitive mode and site of interaction of ticagrelor at the human platelet P2Y12 -receptor.Protease-activated receptor-4 and purinergic receptor P2Y12 dimerize, co-internalize, and activate Akt signaling via endosomal recruitment of β-arrestin.Structure, Pharmacology and Roles in Physiology of the P2Y12 Receptor.Development of 1-Amino-4-(phenylamino)anthraquinone-2-sulfonate Sodium Derivatives as a New Class of Inhibitors of RANKL-Induced Osteoclastogenesis.Structure-Activity Relationships of a Novel Group of Large-Conductance Ca2+-Activated K+(BK) Channel Modulators: The GoSlo-SR Family
P2860
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P2860
High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 receptors.
description
2009 nî lūn-bûn
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2009年の論文
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2009年学术文章
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2009年学术文章
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2009年学术文章
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2009年学术文章
@zh-my
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name
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@en
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@nl
type
label
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@en
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@nl
prefLabel
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@en
High-affinity, non-nucleotide- ...... s of platelet P2Y12 receptors.
@nl
P50
P356
P1476
High-affinity, non-nucleotide-derived competitive antagonists of platelet P2Y12 receptors
@en
P2093
Kerstin Atzler
Markus Glänzel
P304
P356
10.1021/JM9003297
P407
P577
2009-06-01T00:00:00Z