Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
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SuFEx: a metal-free click ligation for multivalent biomolecules.Multidimensional SuFEx Click Chemistry: Sequential Sulfur(VI) Fluoride Exchange Connections of Diverse Modules Launched From An SOF4 Hub.Click chemistry patents and their impact on drug discovery and chemical biology.Cell permeable affinity- and activity-based probes.Arylfluorosulfates Inactivate Intracellular Lipid Binding Protein(s) through Chemoselective SuFEx Reaction with a Binding Site Tyr ResidueRational Design of a Water-Soluble, Lipid-Compatible Fluorescent Probe for Cu(I) with Sub-Part-Per-Trillion Sensitivity.Recent advances in click chemistry applied to dendrimer synthesis.Lysine-Targeting Covalent Inhibitors.Discovery of novel anti-HIV agents via Cu(I)-catalyzed azide-alkyne cycloaddition (CuAAC) click chemistry-based approach.Broad-Spectrum Kinase Profiling in Live Cells with Lysine-Targeted Sulfonyl Fluoride Probes.Sulfonyl fluorides as privileged warheads in chemical biologySynthesis of Sulfotyrosine-Containing Peptides by Incorporating Fluorosulfated Tyrosine Using an Fmoc-Based Solid-Phase Strategy.Reengineering Antibiotics to Combat Bacterial Resistance: Click Chemistry [1,2,3]-Triazole Vancomycin Dimers with Potent Activity against MRSA and VRE.One-pot palladium-catalyzed synthesis of sulfonyl fluorides from aryl bromides.Chemoselective Synthesis of Polysubstituted Pyridines from Heteroaryl Fluorosulfates.Copper(i)-catalyzed sulfonylative Suzuki-Miyaura cross-coupling.Palladium-Catalyzed Fluorosulfonylvinylation of Organic Iodides.A Heck-Matsuda Process for the Synthesis of β-Arylethenesulfonyl Fluorides: Selectively Addressable Bis-electrophiles for SuFEx Click Chemistry.N-Heterocyclic Carbene Catalyzed Synthesis of δ-Sultones via α,β-Unsaturated Sulfonyl Azolium Intermediates.Bifluoride-catalysed sulfur(VI) fluoride exchange reaction for the synthesis of polysulfates and polysulfonates."Inverse Drug Discovery" Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates.Combining Click Sulfur(VI)-Fluoride Exchange with Photoiniferters: A Facile, Fast, and Efficient Strategy for Postpolymerization Modification.A study of the reactivity of S(VI)-F containing warheads with nucleophilic amino-acid side chains under physiological conditions.SuFEx-Based Polysulfonate Formation from Ethenesulfonyl Fluoride-Amine Adducts.SO2 F2 -Mediated One-Pot Synthesis of Aryl Carboxylic Acids and Esters from Phenols through a Pd-Catalyzed Insertion of Carbon Monoxide.Ethenesulfonyl Fluoride: The Most Perfect Michael Acceptor Ever Found?A Vinyl Sulfone-Based Fluorogenic Probe Capable of Selective Labeling of PHGDH in Live Mammalian Cells.SuFEx Click: New Materials from SOx F and Silyl Ethers.Sulfur-Fluoride Exchange (SuFEx)-Mediated Synthesis of Sterically Hindered and Electron-Deficient Secondary and Tertiary Amides via Acyl Fluoride Intermediates.SuFEx Chemistry of Thionyl Tetrafluoride (SOF4 ) with Organolithium Nucleophiles: Synthesis of Sulfonimidoyl Fluorides, Sulfoximines, Sulfonimidamides, and Sulfonimidates.Chemoselective Preparation of Clickable Aryl Sulfonyl Fluoride Monomers: A Toolbox of Highly Functionalized Intermediates for Chemical Biology Probe Synthesis.SuFEx on the Surface: A Flexible Platform for Postpolymerization Modification of Polymer Brushes.Genetically Encoding Fluorosulfate-l-tyrosine To React with Lysine, Histidine, and Tyrosine via SuFEx in Proteins in Vivo.Strain-Promoted Cycloaddition of Cyclopropenes with o-Quinones: A Rapid Click Reaction.Trifluoromethylfluorosulfonylation of Unactivated Alkenes Using Readily Available Ag(O2 CCF2 SO2 F) and N-Fluorobenzenesulfonimide.Aryl Fluorosulfate Trapped Staudinger Reduction.Patent highlights: December 2015-January 2016.Pd(PPh3 )4 -Catalyzed Buchwald-Hartwig Amination ofAryl Fluorosulfonates with Aryl AminesCellular thermal shift and clickable chemical probe assays for the determination of drug-target engagement in live cellsQuantitative and Orthogonal Formation and Reactivity of SuFEx Platforms
P2860
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P2860
Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
description
2014 nî lūn-bûn
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2014年の論文
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2014年学术文章
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2014年学术文章
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2014年学术文章
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2014年学术文章
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2014年學術文章
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name
Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
@en
type
label
Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
@en
prefLabel
Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
@en
P2860
P356
P1476
Sulfur(VI) fluoride exchange (SuFEx): another good reaction for click chemistry.
@en
P2093
Jiajia Dong
Larissa Krasnova
P2860
P304
P356
10.1002/ANIE.201309399
P407
P577
2014-08-11T00:00:00Z