Synthesis and biological evaluation of substituted [18F]imidazo[1,2-a]pyridines and [18F]pyrazolo[1,5-a]pyrimidines for the study of the peripheral benzodiazepine receptor using positron emission tomography.
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Synthesis and biological evaluation of glucagon-like peptide-1 receptor agonists.Towards molecular imaging of multiple sclerosis.A graphical method to compare the in vivo binding potential of PET radioligands in the absence of a reference region: application to [¹¹C]PBR28 and [¹⁸F]PBR111 for TSPO imaging.Fluorinated molecules in the diagnosis and treatment of neurodegenerative diseases.In vivo binding of protoporphyrin IX to rat translocator protein imaged with positron emission tomographyTwo binding sites for [3H]PBR28 in human brain: implications for TSPO PET imaging of neuroinflammation.Biodistribution and radiation dosimetry in humans of a new PET ligand, (18)F-PBR06, to image translocator protein (18 kDa).[18F]FEBMP: Positron Emission Tomography Imaging of TSPO in a Model of Neuroinflammation in Rats, and in vitro Autoradiograms of the Human Brain.Radiosynthesis, In Vivo Biological Evaluation, and Imaging of Brain Lesions with [123I]-CLINME, a New SPECT Tracer for the Translocator ProteinSingle-step high-yield radiosynthesis and evaluation of a sensitive 18F-labeled ligand for imaging brain peripheral benzodiazepine receptors with PET.Imaging microglial activation during neuroinflammation and Alzheimer's disease.Quantification of translocator protein (18 kDa) in the human brain with PET and a novel radioligand, (18)F-PBR06.The potential of carbon-11 and fluorine-18 chemistry: illustration through the development of positron emission tomography radioligands targeting the translocator protein 18 kDa.Alternative approaches for PET radiotracer development in Alzheimer's disease: imaging beyond plaque.Synthesis of imidazo[1,2-a]pyridines: a decade update.Excited-state intramolecular proton-transfer (ESIPT)-inspired solid state emitters.Comparison of in vivo binding properties of the 18-kDa translocator protein (TSPO) ligands [(18)F]PBR102 and [ (18)F]PBR111 in a model of excitotoxin-induced neuroinflammation.PET imaging of brain inflammation during early epileptogenesis in a rat model of temporal lobe epilepsy.Radiosynthesis and Preclinical Evaluation of [18F]F-DPA, A Novel Pyrazolo[1,5a]pyrimidine Acetamide TSPO Radioligand, in Healthy Sprague Dawley RatsGeneral and efficient copper-catalyzed three-component coupling reaction towards imidazoheterocycles: one-pot synthesis of alpidem and zolpidemThe development of an automated and GMP compliant FASTlab™ Synthesis of [(18) F]GE-180; a radiotracer for imaging translocator protein (TSPO).Preparation of imidazo[1,2-a]-N-heterocyclic derivatives with gem-difluorinated side chains.Preclinical in vivo and in vitro comparison of the translocator protein PET ligands [18F]PBR102 and [18F]PBR111.Recent Progress in the Development of TSPO PET Ligands for Neuroinflammation Imaging in Neurological Diseases.[18F]DPA-C5yne, a novel fluorine-18-labelled analogue of DPA-714: radiosynthesis and preliminary evaluation as a radiotracer for imaging neuroinflammation with PET.
P2860
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P2860
Synthesis and biological evaluation of substituted [18F]imidazo[1,2-a]pyridines and [18F]pyrazolo[1,5-a]pyrimidines for the study of the peripheral benzodiazepine receptor using positron emission tomography.
description
2008 nî lūn-bûn
@nan
2008年の論文
@ja
2008年学术文章
@wuu
2008年学术文章
@zh
2008年学术文章
@zh-cn
2008年学术文章
@zh-hans
2008年学术文章
@zh-my
2008年学术文章
@zh-sg
2008年學術文章
@yue
2008年學術文章
@zh-hant
name
Synthesis and biological evalu ...... positron emission tomography.
@en
Synthesis and biological evalu ...... positron emission tomography.
@nl
type
label
Synthesis and biological evalu ...... positron emission tomography.
@en
Synthesis and biological evalu ...... positron emission tomography.
@nl
prefLabel
Synthesis and biological evalu ...... positron emission tomography.
@en
Synthesis and biological evalu ...... positron emission tomography.
@nl
P2093
P356
P1476
Synthesis and biological evalu ...... positron emission tomography.
@en
P2093
Andrew Katsifis
Christian Loc'h
Christopher J R Fookes
Filomena Mattner
Ivan Greguric
Marie-Claude Gregoire
Paula Berghofer
Rachael Shepherd
Tien Q Pham
P304
P356
10.1021/JM7014556
P407
P577
2008-06-17T00:00:00Z