Interaction of convulsive ligands with benzodiazepine receptors.
about
7-Chlorokynurenic acid is a selective antagonist at the glycine modulatory site of the N-methyl-D-aspartate receptor complexThe pharmacological properties of the imidazobenzodiazepine, FG 8205, a novel partial agonist at the benzodiazepine receptorNegative modulation of α₅ GABAA receptors in rats may partially prevent memory impairment induced by MK-801, but not amphetamine- or MK-801-elicited hyperlocomotionReal-time analysis of dopamine: antagonist interactions at recombinant human D2long receptor upon modulation of its activation stateThe affinities, potencies and efficacies of some benzodiazepine-receptor agonists, antagonists and inverse-agonists at rat hippocampal GABAA-receptorsIsolation, characterization, and purification to homogeneity of an endogenous polypeptide with agonistic action on benzodiazepine receptors[11C]flumazenil binding is increased in a dose-dependent manner with tiagabine-induced elevations in GABA levelsBenzodiazepine Receptors and Their Relationship to the Treatment of EpilepsyBeyond classical benzodiazepines: novel therapeutic potential of GABAA receptor subtypes.Inverse agonism at G protein-coupled receptors: (patho)physiological relevance and implications for drug discovery.Ontogenic profile of seizures evoked by the beta-carboline DMCM (methyl-6,7-dimethoxy-4-ethyl-β-carboline-3-carboxylate) in rats.Effects of GABA modulators on the repeated acquisition of response sequences in squirrel monkeys.Benzodiazepines and anterior pituitary function.Inverse agonism and its therapeutic significance.Antagonists with negative intrinsic activity at delta opioid receptors coupled to GTP-binding proteins.Protection against the lethal effects of pentobarbital in mice by a benzodiazepine receptor inverse agonist, 6,7-dimethoxy-4-ethyl-3-carbomethoxy-beta-carboline.Protracted treatment with diazepam increases the turnover of putative endogenous ligands for the benzodiazepine/beta-carboline recognition siteA 7-phenyl substituted triazolopyridazine has inverse agonist activity at the benzodiazepine receptor siteIncrease in the Bmax of gamma-aminobutyric acid-A recognition sites in brain regions of mice receiving diazepam.Putative diazepam binding inhibitor peptide: cDNA clones from rat.Individually monitoring ligand-induced changes in the structure of the GABAA receptor at benzodiazepine binding site and non-binding-site interfaces.Response to diazepam in children with malaria-induced seizures.Tiagabine increases [11C]flumazenil binding in cortical brain regions in healthy control subjectsbeta-Carbolines enhance shock-induced suppression of drinking in rats.Benzodiazepine receptor-mediated enhancement and inhibition of taste reactivity, food choice, and intake.Benzodiazepines.The benzodiazepine receptor.Benzodiazepines in perspective (II): The GABAA-Benzodiazepine Receptor Ligands.[Current hypotheses of the central mechanism of action of benzodiazepine tranquilizers]Interaction of beta-carboline inverse agonists for the benzodiazepine site with another site on GABAA receptors.The effects of benzodiazepine agonists, inverse agonists and Ro 15-1788 on the responses of the superior cervical ganglion to GABA in vitro.Acute and chronic effects of the benzodiazepine receptor ligand FG 7142: proconvulsant properties and kindlingAllosteric modulation of an expressed homo-oligomeric GABA-gated chloride channel of Drosophila melanogasterAgonist-independent activation of Gz by the 5-hydroxytryptamine1A receptor co-expressed in Spodoptera frugiperda cells. Distinguishing inverse agonists from neutral antagonists.Benzodiazepine-induced intestinal motor disturbances in rats: mediation by omega 2 (BZ2) sites on capsaicin-sensitive afferent neuronesInverse agonist activities of beta-adrenoceptor antagonists in rat myocardium.Characterization of [3H]-imidazenil binding to rat brain membranesFunctional importance of the Ala(116)-Pro(136) region in the calcium-sensing receptor. Constitutive activity and inverse agonism in a family C G-protein-coupled receptor.Up-regulation of a constitutively active form of the beta2-adrenoceptor by sustained treatment with inverse agonists but not antagonists.Electrophysiological studies in cultured mouse CNS neurones of the actions of an agonist and an inverse agonist at the benzodiazepine receptor.
P2860
Q24649753-3588F585-B24A-4854-8757-0CB66CE964FBQ24673465-533B0DFA-11DE-4671-8DD6-3A14E95DD848Q27325106-80E80B0D-9EDE-4F75-ADBC-A86BD5ADA059Q28346724-51729848-6BC7-455A-AD03-A605E804468FQ28360605-2D21FC6A-2D95-4A85-B930-B16B6079AEB2Q28568270-28EAAA85-0CF7-4C57-980B-5670DC86ADC9Q28731698-7E0B6006-D3EB-4DE5-AD20-ED0831AB6BB6Q29040772-9B86FEAE-983F-4EBB-BD47-285816122210Q30466591-C66B75DA-C8B2-469F-89D6-FC3B70DCD0E2Q33898777-9AAB14A7-36FE-4BFF-A1B7-AF98C85F8ACFQ34098194-AADE2C58-A49B-46E9-A81D-918703633F15Q34137074-4628FCC0-3A71-438A-A063-BB48282E3186Q34150270-40FDFF0E-FF7D-4C37-BC72-67B1B0C155B6Q34226789-5A04B9C6-F2EF-49C9-985D-1F5C1EC8D0E1Q34306079-74A599E3-42A7-4CAC-BD31-1B9935D29A2BQ34559437-00BFAC51-CD95-4157-81CA-2F7719ED5B87Q34603222-7D80B8F4-535C-4DE7-8B14-AA2DC1FA1383Q35887671-D6A539F8-5EC0-4A08-A8A8-E4DF7D65DAECQ36267603-B3488E09-D97E-41D0-A366-05D6F6CBD204Q36458516-54A43292-C947-40AB-A51E-D166B9668F2FQ36907077-9730C3F8-FE2F-42BB-9494-FADB9CB4FFC4Q37008323-1C8C7DD7-D3B6-4BC3-BEF1-C2652816D60CQ37369444-1ECB1A5A-0C6A-4ED3-8801-8E101466AC06Q37608273-BE9F835B-F907-492F-810D-9FF52A5818B7Q38328766-741E4D28-F1CF-4A17-8B8A-328FECA24CA0Q39180030-E7F9E9C7-D6AD-4491-ADB3-01FD8FCA20D4Q39505550-7098C29B-8A23-4781-A058-805E932B92D8Q40776362-10E09B05-EA65-4C96-A741-7D167E51874FQ41135772-17B8E815-BD60-4B71-A55F-6C453A4528B2Q41364446-B12B3CA9-8C26-4AA1-9887-029243E1927CQ41739206-92E571F1-2B5C-46CF-9EF4-6BDCD24D2FFBQ41744092-3BD4B37B-1FA4-45E9-8780-CBA6CFFFB31DQ41881591-EAAAF3DD-BAB3-4EA0-A249-03758A31AD84Q42061317-E398FF48-89E6-44E5-A102-BF74F8DADB5CQ42090522-8F63B558-CB05-456A-B7C0-D11DA2C4B453Q42123749-7C56FBA6-CF98-421B-AF9F-17D85885E603Q42370041-7E19340F-45E6-454F-BE8F-0916215B35DFQ42488693-CB488300-E844-407D-8E01-081354ECC9BEQ42528493-BC34D695-0338-418E-8AB0-7310576844A3Q42568954-2DADE7BF-65A4-47D0-8866-43E6800B8FE1
P2860
Interaction of convulsive ligands with benzodiazepine receptors.
description
1982 nî lūn-bûn
@nan
1982年の論文
@ja
1982年学术文章
@wuu
1982年学术文章
@zh
1982年学术文章
@zh-cn
1982年学术文章
@zh-hans
1982年学术文章
@zh-my
1982年学术文章
@zh-sg
1982年學術文章
@yue
1982年學術文章
@zh-hant
name
Interaction of convulsive ligands with benzodiazepine receptors.
@en
Interaction of convulsive ligands with benzodiazepine receptors.
@nl
type
label
Interaction of convulsive ligands with benzodiazepine receptors.
@en
Interaction of convulsive ligands with benzodiazepine receptors.
@nl
prefLabel
Interaction of convulsive ligands with benzodiazepine receptors.
@en
Interaction of convulsive ligands with benzodiazepine receptors.
@nl
P2093
P356
P1433
P1476
Interaction of convulsive ligands with benzodiazepine receptors.
@en
P2093
C Braestrup
E N Petersen
R Schmiechen
P304
P356
10.1126/SCIENCE.6281892
P407
P577
1982-06-01T00:00:00Z