Structure-activity relationship study of selective excitatory amino acid transporter subtype 1 (EAAT1) inhibitor 2-amino-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrile (UCPH-101) and absolute configuratio
about
Mechanisms of glutamate transportSLC transporters as therapeutic targets: emerging opportunitiesβ-amino esters from the reductive ring opening of aziridine-2-carboxylates.Structure-activity-relationship study of N-acyl-N-phenylpiperazines as potential inhibitors of the Excitatory Amino Acid Transporters (EAATs): improving the potency of a micromolar screening Hit is not truism.SLC1 glutamate transportersProbing for improved potency and in vivo bioavailability of excitatory amino acid transporter subtype 1 inhibitors UCPH-101 and UCPH-102: design, synthesis and pharmacological evaluation of substituted 7-biphenyl analogs.Vibrational circular dichroism discrimination of diastereomeric cedranol acetates.Depression following traumatic brain injury in mice is associated with down-regulation of hippocampal astrocyte glutamate transporters by thrombin.Bioavailability Studies and in vitro Profiling of the Selective Excitatory Amino Acid Transporter Subtype 1 (EAAT1) Inhibitor UCPH-102.
P2860
Q26830761-74C09ED6-2B14-46ED-BEB3-26A18EE9EC53Q27014726-D4E18C6C-890A-41BB-A66F-16FCD08633A1Q34488638-088A9F9E-E9BE-412C-B4C7-FA47D200E482Q35532022-16E5492A-9BCD-4517-BEEA-7D4C518078BDQ37495425-3AA4705A-CA8E-4030-A680-39DB447B4FFCQ39219745-4F909DB0-F3FB-489F-8D1B-56341AAAC9CEQ44428017-43B10EC4-A832-4655-A947-F01FBAFDE12FQ47709165-DED31D36-C434-4A10-B94D-1EB7E638CE3EQ48956786-6DBF7D0C-6F6D-455B-A269-69783BAEEB0C
P2860
Structure-activity relationship study of selective excitatory amino acid transporter subtype 1 (EAAT1) inhibitor 2-amino-4-(4-methoxyphenyl)-7-(naphthalen-1-yl)-5-oxo-5,6,7,8-tetrahydro-4H-chromene-3-carbonitrile (UCPH-101) and absolute configuratio
description
2012 nî lūn-bûn
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2012年の論文
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2012年学术文章
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2012年学术文章
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2012年学术文章
@zh-cn
2012年学术文章
@zh-hans
2012年学术文章
@zh-my
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2012年學術文章
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name
Structure-activity relationshi ...... 101) and absolute configuratio
@en
Structure-activity relationshi ...... 101) and absolute configuratio
@nl
type
label
Structure-activity relationshi ...... 101) and absolute configuratio
@en
Structure-activity relationshi ...... 101) and absolute configuratio
@nl
prefLabel
Structure-activity relationshi ...... 101) and absolute configuratio
@en
Structure-activity relationshi ...... 101) and absolute configuratio
@nl
P2093
P50
P356
P1476
Structure-activity relationshi ...... itio Hartree-Fock calculations
@en
P2093
Bjarke Abrahamsen
Henrik Bohr
Irene Shim
Tri H V Huynh
P304
P356
10.1021/JM300345Z
P407
P577
2012-05-17T00:00:00Z