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Q38821763-8193C494-8C82-4CE3-90F1-C490E6245242
Q38821763-8193C494-8C82-4CE3-90F1-C490E6245242
BestRank
Statement
http://www.wikidata.org/entity/statement/Q38821763-8193C494-8C82-4CE3-90F1-C490E6245242
Modular Assembly of Allosteric MEK Inhibitor Structural Elements Unravels Potency and Feedback-Modulation Handles.
P2860
Q38821763-8193C494-8C82-4CE3-90F1-C490E6245242
BestRank
Statement
http://www.wikidata.org/entity/statement/Q38821763-8193C494-8C82-4CE3-90F1-C490E6245242
rank
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Statement
wasDerivedFrom
a02ed6d230e5c35b95b6e64945fe7f136096daed
P2860
The sulfamide moiety affords higher inhibitory activity and oral bioavailability to a series of coumarin dual selective RAF/MEK inhibitors.