Artemisinin and a Series of Novel Endoperoxide Antimalarials Exert Early Effects on Digestive Vacuole Morphology
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A plausible mechanism for the antimalarial activity of artemisinin: A computational approachArtemisinin-based combination therapies: a vital tool in efforts to eliminate malariaArtemisinin Action and Resistance in Plasmodium falciparumPlatelet factor 4 activity against P. falciparum and its translation to nonpeptidic mimics as antimalarialsIn vitro sensitivity of Plasmodium falciparum from China-Myanmar border area to major ACT drugs and polymorphisms in potential target genesHit-to-lead development of the chamigrane endoperoxide merulin A for the treatment of African sleeping sicknessReal-time imaging of the intracellular glutathione redox potential in the malaria parasite Plasmodium falciparumCryo transmission X-ray imaging of the malaria parasite, P. falciparum.Dynamic RNA profiling in Plasmodium falciparum synchronized blood stages exposed to lethal doses of artesunate.Artemisinin directly targets malarial mitochondria through its specific mitochondrial activation.Loss of pH control in Plasmodium falciparum parasites subjected to oxidative stress.Mitochondrial metabolism of sexual and asexual blood stages of the malaria parasite Plasmodium falciparum.Tracking Glideosome-associated protein 50 reveals the development and organization of the inner membrane complex of Plasmodium falciparum.Antitumor activity of artemisinin and its derivatives: from a well-known antimalarial agent to a potential anticancer drugInvestigating the antimalarial action of 1,2,4-trioxolanes with fluorescent chemical probesMutations in the Plasmodium falciparum chloroquine resistance transporter, PfCRT, enlarge the parasite's food vacuole and alter drug sensitivities.Mechanisms of in vitro resistance to dihydroartemisinin in Plasmodium falciparum.Monoclonal Antibodies That Recognize the Alkylation Signature of Antimalarial Ozonides OZ277 (Arterolane) and OZ439 (Artefenomel).Artemisinin resistance in rodent malaria--mutation in the AP2 adaptor μ-chain suggests involvement of endocytosis and membrane protein trafficking.Accumulation of artemisinin trioxane derivatives within neutral lipids of Plasmodium falciparum malaria parasites is endoperoxide-dependent.Antimalarials and the fight against malaria in BrazilOrganism-like formation of Schistosoma hemozoin and its function suggest a mechanism for anti-malarial action of artemisinin.In vitro activity of anti-malarial ozonides against an artemisinin-resistant isolate.The pharmacogenetics of antimalaria artemisinin combination therapy.Emerging drugs for malaria.Synthesis of five- and six-membered cyclic organic peroxides: Key transformations into peroxide ring-retaining products.Rapid kill of malaria parasites by artemisinin and semi-synthetic endoperoxides involves ROS-dependent depolarization of the membrane potentialHonoring antiparasitics: The 2015 Nobel Prize in Physiology or Medicine.Probing the antimalarial mechanism of artemisinin and OZ277 (arterolane) with nonperoxidic isosteres and nitroxyl radicals.Phenotypic approach artemisinin resistance in malaria rodent as in vivo model.Enzymes Involved in Pyrophosphate and Calcium Metabolism as Targets for Anti-scuticociliate Chemotherapy.Investigations into the role of the Plasmodium falciparum SERCA (PfATP6) L263E mutation in artemisinin action and resistance.Interactions between artemisinins and other antimalarial drugs in relation to the cofactor model--a unifying proposal for drug action.5-Bromo-spiro-[1,2-dioxane-4,4'-tricyclo-[4.3.1.1]undeca-ne]-3'-ol.In vitro interaction of artemisinin derivatives or the fully synthetic peroxidic anti-malarial OZ277 with thapsigargin in Plasmodium falciparum strains.Induction of high tolerance to artemisinin by sub-lethal administration: A new in vitro model of P. falciparum.Potential of sustainable hierarchical zeolites in the valorization of α-pinene.Targeting Channels and Transporters in Protozoan Parasite Infections.Novel dihydroartemisinin derivative DHA-37 induces autophagic cell death through upregulation of HMGB1 in A549 cells
P2860
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P2860
Artemisinin and a Series of Novel Endoperoxide Antimalarials Exert Early Effects on Digestive Vacuole Morphology
description
2007 nî lūn-bûn
@nan
2007年の論文
@ja
2007年論文
@yue
2007年論文
@zh-hant
2007年論文
@zh-hk
2007年論文
@zh-mo
2007年論文
@zh-tw
2007年论文
@wuu
2007年论文
@zh
2007年论文
@zh-cn
name
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@ast
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en-gb
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@nl
type
label
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@ast
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en-gb
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@nl
altLabel
Artemisinin and a series of no ...... n digestive vacuole morphology
@en
prefLabel
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@ast
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@en-gb
Artemisinin and a Series of No ...... n Digestive Vacuole Morphology
@nl
P2093
P2860
P921
P3181
P356
P1476
Artemisinin and a series of no ...... n digestive vacuole morphology
@en
P2093
Dennis K Taylor
Leann Tilley
Maria del Pilar Crespo
Peter Valente
Tony V Robinson
P2860
P304
P3181
P356
10.1128/AAC.00609-07
P407
P577
2007-10-15T00:00:00Z