Kinetic and Structural Analysis of Bisubstrate Inhibition of the Salmonella enterica Aminoglycoside 6‘- N -Acetyltransferase † , ‡
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Structure and Functional Diversity of GCN5-Related N-Acetyltransferases (GNAT)Strategies to overcome the action of aminoglycoside-modifying enzymes for treating resistant bacterial infectionsProtein lysine acetylation by p300/CBPCrystal structure of RimI fromSalmonella typhimurium LT2, the GNAT responsible for Nα-acetylation of ribosomal protein S18Structure of the complex of Neisseria gonorrhoeae N-acetyl-l-glutamate synthase with a bound bisubstrate analogAminoglycoside modifying enzymes.Synthesis of a phosphonate-linked aminoglycoside-coenzyme a bisubstrate and use in mechanistic studies of an enzyme involved in aminoglycoside resistanceIdentification of an Inhibitor of the Aminoglycoside 6'-N-Acetyltransferase type Ib [AAC(6')-Ib] by Glide Molecular DockingCosubstrate tolerance of the aminoglycoside resistance enzyme Eis from Mycobacterium tuberculosisRise and dissemination of aminoglycoside resistance: the aac(6')-Ib paradigm.Inhibitors of aminoglycoside resistance activated in cells.Understanding and overcoming aminoglycoside resistance caused by N-6'-acetyltransferase.Global ITC fitting methods in studies of protein allostery.Effects of altering aminoglycoside structures on bacterial resistance enzyme activities.The RimL transacetylase provides resistance to translation inhibitor microcin CMultiple keys for a single lock: the unusual structural plasticity of the nucleotidyltransferase (4')/kanamycin complex.
P2860
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P2860
Kinetic and Structural Analysis of Bisubstrate Inhibition of the Salmonella enterica Aminoglycoside 6‘- N -Acetyltransferase † , ‡
description
2008 nî lūn-bûn
@nan
2008 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@ast
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@en
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@nl
type
label
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@ast
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@en
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@nl
prefLabel
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@ast
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@en
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@nl
P2093
P2860
P3181
P356
P1433
P1476
Kinetic and Structural Analysi ...... 6‘- N -Acetyltransferase † , ‡
@en
P2093
John S Blanchard
Karine Auclair
Lee Freiburger
Maria L B Magalhães
Matthew W Vetting
P2860
P304
P3181
P356
10.1021/BI701957C
P407
P577
2008-01-15T00:00:00Z