The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
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ROR nuclear receptors: structures, related diseases, and drug discoveryIvermectin - Old Drug, New Tricks?An antagonist of the retinoid X receptor reduces the viability of Trichuris muris in vitroCoordinated Actions of FXR and LXR in Metabolism: From Pathogenesis to Pharmacological Targets for Type 2 DiabetesRecent advances in the understanding and management of rosacea.The river blindness drug Ivermectin and related macrocyclic lactones inhibit WNT-TCF pathway responses in human cancer.Structural Basis for Small Molecule NDB (N-Benzyl-N-(3-(tert-butyl)-4-hydroxyphenyl)-2,6-dichloro-4-(dimethylamino) Benzamide) as a Selective Antagonist of Farnesoid X Receptor α (FXRα) in Stabilizing the Homodimerization of the Receptor.Selective targeting of nuclear receptor FXR by avermectin analogues with therapeutic effects on nonalcoholic fatty liver disease.Quantitative high-throughput profiling of environmental chemicals and drugs that modulate farnesoid X receptorTargeting nuclear receptors with marine natural products.Topical ivermectin improves allergic skin inflammation.Inhibition of Plasmodium Liver Infection by Ivermectin.Bioenergetic cues shift FXR splicing towards FXRα2 to modulate hepatic lipolysis and fatty acid metabolism.On the relationship of anthranilic derivatives structure and the FXR (Farnesoid X receptor) agonist activity.Ivermectin and its target molecules: shared and unique modulation mechanisms of ion channels and receptors by ivermectin.Ivermectin activates GIRK channels in a PIP2 -dependent, Gβγ -independent manner and an amino acid residue at the slide helix governs the activation.Repurposed FDA-approved drugs targeting genes influencing aging can extend lifespan and healthspan in rotifers.Differential modulation of FXR activity by chlorophacinone and ivermectin analogs.Discovery of new non-steroidal farnesoid X receptor modulators through 3D shape similarity search and structure-based virtual screening.Discovery of Natural Products as Novel and Potent FXR Antagonists by Virtual Screening.Structural insights into the heterodimeric complex of the nuclear receptors FXR and RXR
P2860
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P2860
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
description
2013 nî lūn-bûn
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2013 թուականին հրատարակուած գիտական յօդուած
@hyw
2013 թվականին հրատարակված գիտական հոդված
@hy
2013年の論文
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2013年論文
@yue
2013年論文
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2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
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name
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@ast
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@en
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@nl
type
label
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@ast
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@en
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@nl
prefLabel
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@ast
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@en
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@nl
P2093
P2860
P356
P1476
The antiparasitic drug ivermectin is a novel FXR ligand that regulates metabolism
@en
P2093
Hongyan Liu
Shanshan Wang
Shengchen Lin
Weili Zheng
P2860
P2888
P356
10.1038/NCOMMS2924
P407
P577
2013-01-01T00:00:00Z
P5875
P6179
1043683656