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Jump into a New Fold-A Homology Based Model for the ABCG2/BCRP Multidrug TransporterTransmembrane helices 1 and 6 of the human breast cancer resistance protein (BCRP/ABCG2): identification of polar residues important for drug transport.Mutational analysis of threonine 402 adjacent to the GXXXG dimerization motif in transmembrane segment 1 of ABCG2.Role of basic residues within or near the predicted transmembrane helix 2 of the human breast cancer resistance protein in drug transport.Structure and function of the human breast cancer resistance protein (BCRP/ABCG2).The challenge of exploiting ABCG2 in the clinic.Structure and function of BCRP, a broad specificity transporter of xenobiotics and endobiotics.Identification of residues in ABCG2 affecting protein trafficking and drug transport, using co-evolutionary analysis of ABCG sequences.Mutation of Glu521 or Glu535 in cytoplasmic loop 5 causes differential misfolding in multiple domains of multidrug and organic anion transporter MRP1 (ABCC1)Posttranslational negative regulation of glycosylated and non-glycosylated BCRP expression by Derlin-1.The structure of the human ABC transporter ABCG2 reveals a novel mechanism for drug extrusion.Clinically relevant mutations in the ABCG2 transporter uncovered by genetic analysis linked to erythrocyte membrane protein expression.
P2860
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P2860
description
2009 nî lūn-bûn
@nan
2009 թուականի Մայիսին հրատարակուած գիտական յօդուած
@hyw
2009 թվականի մայիսին հրատարակված գիտական հոդված
@hy
2009年の論文
@ja
2009年学术文章
@wuu
2009年学术文章
@zh-cn
2009年学术文章
@zh-hans
2009年学术文章
@zh-my
2009年学术文章
@zh-sg
2009年學術文章
@yue
name
Arginine 383 is a crucial residue in ABCG2 biogenesis
@ast
Arginine 383 is a crucial residue in ABCG2 biogenesis
@en
Arginine 383 is a crucial residue in ABCG2 biogenesis
@nl
type
label
Arginine 383 is a crucial residue in ABCG2 biogenesis
@ast
Arginine 383 is a crucial residue in ABCG2 biogenesis
@en
Arginine 383 is a crucial residue in ABCG2 biogenesis
@nl
prefLabel
Arginine 383 is a crucial residue in ABCG2 biogenesis
@ast
Arginine 383 is a crucial residue in ABCG2 biogenesis
@en
Arginine 383 is a crucial residue in ABCG2 biogenesis
@nl
P2093
P2860
P50
P1476
Arginine 383 is a crucial residue in ABCG2 biogenesis
@en
P2093
Ajay Sharma
Balazs Sarkadi
Csilla Ozvegy-Laczka
Lilangi S Ediriwickrema
Orsolya Polgar
Susan E Bates
Yvona Ward
P2860
P304
P356
10.1016/J.BBAMEM.2009.04.016
P407
P577
2009-05-03T00:00:00Z