Morphine-induced receptor endocytosis in a novel knockin mouse reduces tolerance and dependence.
about
Opioid receptors: toward separation of analgesic from undesirable effectsAnti-analgesic effect of the mu/delta opioid receptor heteromer revealed by ligand-biased antagonismEndocytosis and signalling: intertwining molecular networksIdentification of the First Marine-Derived Opioid Receptor "Balanced" Agonist with a Signaling Profile That Resembles the EndorphinsBiomarkers of morphine tolerance and dependence are prevented by morphine-induced endocytosis of a mutant mu-opioid receptor.Chronic ethanol consumption in rats produces opioid antinociceptive tolerance through inhibition of mu opioid receptor endocytosis.Opioid-receptor-heteromer-specific trafficking and pharmacology.micro-Opioid receptor endocytosis prevents adaptations in ventral tegmental area GABA transmission induced during naloxone-precipitated morphine withdrawal.How to design an opioid drug that causes reduced tolerance and dependence.Rapid delivery of internalized signaling receptors to the somatodendritic surface by sequence-specific local insertion.Ligand-directed trafficking of the δ-opioid receptor in vivo: two paths toward analgesic tolerance.The role of beta-arrestin2 in the severity of antinociceptive tolerance and physical dependence induced by different opioid pain therapeutics.Examining the role of mu opioid receptor endocytosis in the beneficial and side-effects of prolonged opioid use: from a symposium on new concepts in mu-opioid pharmacologyFunctionally selective signaling for morphine and fentanyl antinociception and tolerance mediated by the rat periaqueductal gray.Opioid receptor desensitization: mechanisms and its link to toleranceChange in functional selectivity of morphine with the development of antinociceptive tolerance.Prolonged morphine treatment alters δ opioid receptor post-internalization traffickingA novel knock-in mouse reveals mechanistically distinct forms of morphine tolerance.The delta opioid receptor: an evolving target for the treatment of brain disorders.Chronic methadone treatment shows a better cost/benefit ratio than chronic morphine in mice.Opioid receptor internalization contributes to dermorphin-mediated antinociceptionMechanisms of rapid opioid receptor desensitization, resensitization and tolerance in brain neurons.Ligand-directed signalling within the opioid receptor family.Regulation of μ-opioid receptors: desensitization, phosphorylation, internalization, and tolerance.Role of ubiquitination in endocytic trafficking of G-protein-coupled receptors.Quantitative encoding of the effect of a partial agonist on individual opioid receptors by multisite phosphorylation and threshold detection.Opioid-Induced GABA potentiation after chronic morphine attenuates the rewarding effects of opioids in the ventral tegmental area.Divergent modes for cargo-mediated control of clathrin-coated pit dynamicsIn vivo trafficking of endogenous opioid receptors.Functional characterization of human variants of the mu-opioid receptor geneRegulation of opioid receptors by endocytic membrane traffic: mechanisms and translational implications.Regulation of opioid receptor signalling: implications for the development of analgesic tolerance.Opioid receptor trafficking and signaling: what happens after opioid receptor activation?Evidence from basic research for opioid combinations.Molecular Perspectives for mu/delta Opioid Receptor Heteromers as Distinct, Functional ReceptorsParadoxical relationship between RAVE (relative activity versus endocytosis) values of several opioid receptor agonists and their liability to cause dependence.Morphine-like opiates selectively antagonize receptor-arrestin interactions.Alternative splicing determines the post-endocytic sorting fate of G-protein-coupled receptors.An immunocytochemical-derived correlate for evaluating the bridging of heteromeric mu-delta opioid protomers by bivalent ligands.The doctor's dilemma: opiate analgesics and chronic pain.
P2860
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P2860
Morphine-induced receptor endocytosis in a novel knockin mouse reduces tolerance and dependence.
description
2008 nî lūn-bûn
@nan
2008 թուականի Յունուարին հրատարակուած գիտական յօդուած
@hyw
2008 թվականի հունվարին հրատարակված գիտական հոդված
@hy
2008年の論文
@ja
2008年論文
@yue
2008年論文
@zh-hant
2008年論文
@zh-hk
2008年論文
@zh-mo
2008年論文
@zh-tw
2008年论文
@wuu
name
Morphine-induced receptor endo ...... uces tolerance and dependence.
@ast
Morphine-induced receptor endo ...... uces tolerance and dependence.
@en
Morphine-induced receptor endo ...... uces tolerance and dependence.
@nl
type
label
Morphine-induced receptor endo ...... uces tolerance and dependence.
@ast
Morphine-induced receptor endo ...... uces tolerance and dependence.
@en
Morphine-induced receptor endo ...... uces tolerance and dependence.
@nl
prefLabel
Morphine-induced receptor endo ...... uces tolerance and dependence.
@ast
Morphine-induced receptor endo ...... uces tolerance and dependence.
@en
Morphine-induced receptor endo ...... uces tolerance and dependence.
@nl
P2093
P2860
P1433
P1476
Morphine-induced receptor endo ...... uces tolerance and dependence.
@en
P2093
Amy M Chang
Carsten K Nielsen
Chrissi J Ou
Dragana Cado
Jennifer L Whistler
Joseph A Kim
Madeline Ferwerda
Maria Waldhoer
Selena Bartlett
P2860
P304
P356
10.1016/J.CUB.2007.12.057
P407
P577
2008-01-01T00:00:00Z