Regulation of μ-opioid receptors: desensitization, phosphorylation, internalization, and tolerance.
about
The search for novel analgesics: targets and mechanismsNeurobiology of opioid dependence in creating addiction vulnerabilityOpioid-induced constipation: advances and clinical guidancePain and Poppies: The Good, the Bad, and the Ugly of Opioid AnalgesicsNovel GPCR paradigms at the μ-opioid receptorPositive allosteric modulators of the μ-opioid receptor: a novel approach for future pain medicationsEndocytosis as a biological response in receptor pharmacology: evaluation by fluorescence microscopyCell-autonomous regulation of Mu-opioid receptor recycling by substance P.Dual-Acting Compounds Targeting Endocannabinoid and Endovanilloid Systems-A Novel Treatment Option for Chronic Pain ManagementThe Relationship Between the Mechanisms of Action and Safety Profiles of Intrathecal Morphine and Ziconotide: A Review of the LiteratureMu opioid receptors on primary afferent nav1.8 neurons contribute to opiate-induced analgesia: insight from conditional knockout miceOn the modularity of the intrinsic flexibility of the µ opioid receptor: a computational studyDeficits in neuronal cytochrome P450 activity attenuate opioid analgesia but not opioid side effects.Significance of neuronal cytochrome P450 activity in opioid-mediated stress-induced analgesia.It's MORe exciting than mu: crosstalk between mu opioid receptors and glutamatergic transmission in the mesolimbic dopamine system.The Concise Guide to PHARMACOLOGY 2013/14: G protein-coupled receptorsProcess Pharmacology: A Pharmacological Data Science Approach to Drug Development and TherapyMolecular Signature That Determines the Acute Tolerance of G Protein-Coupled ReceptorsAcute morphine alters GABAergic transmission in the central amygdala during naloxone-precipitated morphine withdrawal: role of cyclic AMP.Desensitization of functional µ-opioid receptors increases agonist off-rate.Upregulation of miR-375 level ameliorates morphine analgesic tolerance in mouse dorsal root ganglia by inhibiting the JAK2/STAT3 pathway.Angiotensin receptor type 1 and endothelin receptor type A on immune cells mediate migration and the expression of IL-8 and CCL18 when stimulated by autoantibodies from systemic sclerosis patientsMolecular signatures of mouse TRPV1-lineage neurons revealed by RNA-Seq transcriptome analysis.Separate GABA afferents to dopamine neurons mediate acute action of opioids, development of tolerance, and expression of withdrawal.Opioid receptor function is regulated by post-endocytic peptide processing.Contribution of adenylyl cyclase modulation of pre- and postsynaptic GABA neurotransmission to morphine antinociception and tolerance.β-arrestin-2-biased agonism of delta opioid receptors sensitizes transient receptor potential vanilloid type 1 (TRPV1) in primary sensory neurons.CB2 Cannabinoid receptors as a therapeutic target-what does the future hold?The role of the blood-brain barrier in the development and treatment of migraine and other pain disorders.Heterologous regulation of Mu-opioid (MOP) receptor mobility in the membrane of SH-SY5Y cells.Opioid-induced mitogen-activated protein kinase signaling in rat enteric neurons following chronic morphine treatment.Amylin receptor signaling in the nucleus accumbens negatively modulates μ-opioid-driven feeding.Morphine drives internal ribosome entry site-mediated hnRNP K translation in neurons through opioid receptor-dependent signaling.Identification and functional characterization of the phosphorylation sites of the neuropeptide FF2 receptor.Alteration of the mu opioid receptor: Ca2+ channel signaling pathway in a subset of rat sensory neurons following chronic femoral artery occlusion.Opioid receptor desensitization: mechanisms and its link to toleranceStabilization of morphine tolerance with long-term dosing: association with selective upregulation of mu-opioid receptor splice variant mRNAs.Cellular signalling of non-synonymous single-nucleotide polymorphisms of the human μ-opioid receptor (OPRM1)Analgesic synergy between opioid and α2 -adrenoceptorsRecent advances on the δ opioid receptor: from trafficking to function.
P2860
Q24288817-E5AB3BB9-3BDD-48C8-90FF-B27846E3FD02Q26742048-F2A421AD-8879-417E-86A6-481AFFE29A25Q26765571-86F856D2-543D-4343-B0BA-84BE18CC600FQ26782928-402E54BE-149C-4E6C-A6B4-4F4A6712B1E2Q26864286-6932830C-DA57-4786-A779-A9F32A59A7C6Q27027736-7F23D24B-D475-49E5-A177-E0610F4D5FD0Q27310207-BD63ECBF-BE03-4C7F-9DF4-0DC1BCD75F8EQ27320979-4A251DCF-981D-4E64-82BD-FD1DED8E8F00Q28067493-06307A6C-90DF-4DAE-BD00-B8485954367AQ28085351-E3F852AD-2AD3-42AF-99EC-C253CA2212F4Q28533332-2E961A1D-91F3-463A-90E0-73CA7386A3EBQ28542919-C7DC8C25-4C1C-47CA-9EE0-C60F48847F7CQ30370517-CD82CB0F-DE37-43EA-A5B3-C1DF6304A061Q30371265-CB75875F-0E04-4F60-BE30-4F6B3FA25D56Q30437184-9C5A3185-B8F1-4B7F-93FB-39484A6A4B39Q30486707-90D29F92-A2DE-4B5C-A639-07A11526C4B8Q31074800-5732BF94-CF3F-4B96-957F-B832CEF149D6Q33655870-3BBF6CC2-11E0-4843-BE52-E1CF24C745BFQ33709318-45AABADE-0189-481A-AEA3-A3CDB860434FQ33742761-955F8ECA-0E33-427E-A356-45E2A0768002Q33758527-A4AF5A25-CB33-429D-AA6D-182896E33149Q33765684-5CE0FB14-3AFF-48CE-896C-B29BCD91C0E1Q33792431-8EA410D4-0785-4903-9EB0-76E165375A0EQ33811040-917561A2-D3CA-453F-8927-456FB19ADD55Q33888590-6D7B56E9-9F55-4AAF-BB10-8135E1A6ADB5Q33923596-5F5A6760-63E0-40EF-A8F8-1A90433F876AQ34039598-4E113413-CB94-42D2-A139-5147D43C3BBEQ34186015-BEB96389-077E-4837-A2AD-525F04B39342Q34304978-9781D22B-950F-4A02-BB1B-362B76DCD3C7Q34317508-33D1DBE8-9DB2-4F2B-B0C2-47449DAF4637Q34323667-910EBFC2-1682-407E-8AC7-A25102D588E0Q34499302-BF67EDDC-80D4-47EF-931D-C3A1371FEEE7Q34579669-D3B7F432-7B25-4F23-9A72-628449EAC443Q34634103-5DD216AF-20D4-4500-AAB5-DA742A46DF65Q34726976-61BDDC28-54A2-4292-966E-004A90475F4BQ34729984-1239C3A9-E918-4278-BEB5-B80659947790Q34926300-6069E924-2FFF-4544-B0A8-6F3A5DD4ECD6Q34939590-82449FA9-3D5E-49EF-9CF8-09C6321AC2C6Q34939644-8A42F094-B5C4-44BA-93E4-9891BAC360BAQ34939664-FE8A89C1-B56A-44F2-A98B-62EDFD4AFEAD
P2860
Regulation of μ-opioid receptors: desensitization, phosphorylation, internalization, and tolerance.
description
2013 nî lūn-bûn
@nan
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
2013年论文
@zh
2013年论文
@zh-cn
name
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@ast
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@en
type
label
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@ast
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@en
prefLabel
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@ast
Regulation of μ-opioid recepto ...... nternalization, and tolerance.
@en
P2093
P2860
P50
P356
P1476
Regulation of μ-opioid recepto ...... internalization, and tolerance
@en
P2093
Charles Chavkin
Christopher J Evans
John T Williams
Macdonald J Christie
Susan L Ingram
Thomas Koch
P2860
P304
P356
10.1124/PR.112.005942
P577
2013-01-15T00:00:00Z