Monoamine transporter and receptor interaction profiles of a new series of designer cathinones.
about
Legal highs: staying on top of the flood of novel psychoactive substancesIntravenous self-administration of entactogen-class stimulants in male ratsSynthetic cathinones and their rewarding and reinforcing effects in rodents.A Fatal Case of Pentedrone and α-Pyrrolidinovalerophenone Poisoning.Pharmacological profile of novel psychoactive benzofurans.The new stimulant designer compound pentedrone exhibits rewarding properties and affects dopaminergic activity.Baths salts, spice, and related designer drugs: the science behind the headlines.The new psychoactive substances 5-(2-aminopropyl)indole (5-IT) and 6-(2-aminopropyl)indole (6-IT) interact with monoamine transporters in brain tissue.Intravenous self-administration of mephedrone, methylone and MDMA in female rats.Discriminative and locomotor effects of five synthetic cathinones in rats and miceDiscriminative-stimulus effects of second generation synthetic cathinones in methamphetamine-trained ratsEffects of α-pyrrolidinopentiophenone and 4-methyl-N-ethylcathinone, two synthetic cathinones commonly found in second-generation "bath salts," on intracranial self-stimulation thresholds in rats.Psychostimulants and movement disorders.Quantitative structure-activity relationship analysis of the pharmacology of para-substituted methcathinone analogues.In vivo potency and efficacy of the novel cathinone α-pyrrolidinopentiophenone and 3,4-methylenedioxypyrovalerone: self-administration and locomotor stimulation in male ratsEffect of Some Psychoactive Drugs Used as 'Legal Highs' on Brain NeurotransmittersThe Effects of 4-Methylethcathinone on Conditioned Place Preference, Locomotor Sensitization, and Anxiety-Like Behavior: A Comparison with Methamphetamine.Effects of MDMA on body temperature in humansN-Alkylated Analogs of 4-Methylamphetamine (4-MA) Differentially Affect Monoamine Transporters and Abuse Liability.Synthetic cathinone pharmacokinetics, analytical methods, and toxicological findings from human performance and postmortem cases.Reporting Two Fatalities Associated with the Use of 4-Methylethcathinone (4-MEC) and a Review of the Literature.Electrophysiological Actions of Synthetic Cathinones on Monoamine Transporters.Predicting the Abuse Liability of Entactogen-Class, New and Emerging Psychoactive Substances via Preclinical Models of Drug Self-administration.Patterns of use and toxicity of new para-halogenated substituted cathinones: 4-CMC (clephedrone), 4-CEC (4-chloroethcatinone) and 4-BMC (brephedrone).'Second-generation' mephedrone analogs, 4-MEC and 4-MePPP, differentially affect monoamine transporter function.Interactions of Cathinone NPS with Human Transporters and Receptors in Transfected Cells.Editor's Highlight: Characterization of Hepatotoxicity Mechanisms Triggered by Designer Cathinone Drugs (β-Keto Amphetamines).Locomotor, discriminative stimulus, and place conditioning effects of MDAI in rodentsIn Vitro Characterization of Psychoactive Substances at Rat, Mouse, and Human Trace Amine-Associated Receptor 1.Locomotor and reinforcing effects of pentedrone, pentylone and methylone in rats.Opioid-induced inhibition of the human 5-HT and noradrenaline transporters in vitro: link to clinical reports of serotonin syndrome.Intended and unintended use of cathinone mixtures.Acute recreational drug toxicity: Comparison of self-reports and results of immunoassay and additional analytical methods in a multicenter European case series."Ecstasy" to addiction: Mechanisms and reinforcing effects of three synthetic cathinone analogs of MDMA.Self-administration and behavioral economics of second-generation synthetic cathinones in male rats.Structure-Activity Relationships of Substituted Cathinones, with Transporter Binding, Uptake, and Release.
P2860
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P2860
Monoamine transporter and receptor interaction profiles of a new series of designer cathinones.
description
2013 nî lūn-bûn
@nan
2013 թուականի Նոյեմբերին հրատարակուած գիտական յօդուած
@hyw
2013 թվականի նոյեմբերին հրատարակված գիտական հոդված
@hy
2013年の論文
@ja
2013年論文
@yue
2013年論文
@zh-hant
2013年論文
@zh-hk
2013年論文
@zh-mo
2013年論文
@zh-tw
2013年论文
@wuu
name
Monoamine transporter and rece ...... series of designer cathinones.
@ast
Monoamine transporter and rece ...... series of designer cathinones.
@en
Monoamine transporter and rece ...... series of designer cathinones.
@nl
type
label
Monoamine transporter and rece ...... series of designer cathinones.
@ast
Monoamine transporter and rece ...... series of designer cathinones.
@en
Monoamine transporter and rece ...... series of designer cathinones.
@nl
prefLabel
Monoamine transporter and rece ...... series of designer cathinones.
@ast
Monoamine transporter and rece ...... series of designer cathinones.
@en
Monoamine transporter and rece ...... series of designer cathinones.
@nl
P1433
P1476
Monoamine transporter and rece ...... series of designer cathinones
@en
P2093
P304
P356
10.1016/J.NEUROPHARM.2013.11.008
P577
2013-11-22T00:00:00Z