Dictyostelium discoideum expresses a malaria chloroquine resistance mechanism upon transfection with mutant, but not wild-type, Plasmodium falciparum transporter PfCRT.
about
PfCRT and its role in antimalarial drug resistanceGenome-wide compensatory changes accompany drug- selected mutations in the Plasmodium falciparum crt geneIdentification of a mutant PfCRT-mediated chloroquine tolerance phenotype in Plasmodium falciparumFunctional characterization of the Plasmodium falciparum chloroquine-resistance transporter (PfCRT) in transformed Dictyostelium discoideum vesiclesMolecular Mechanisms for Drug Hypersensitivity Induced by the Malaria Parasite's Chloroquine Resistance TransporterInvestigation of the Plasmodium falciparum food vacuole through inducible expression of the chloroquine resistance transporter (PfCRT)Glutathione transport: a new role for PfCRT in chloroquine resistanceChloroquine transport via the malaria parasite's chloroquine resistance transporterMultiple drugs compete for transport via the Plasmodium falciparum chloroquine resistance transporter at distinct but interdependent sitesGeographic patterns of Plasmodium falciparum drug resistance distinguished by differential responses to amodiaquine and chloroquineChloroquine-resistant isoforms of the Plasmodium falciparum chloroquine resistance transporter acidify lysosomal pH in HEK293 cells more than chloroquine-sensitive isoforms.Characterization of the chloroquine resistance transporter homologue in Toxoplasma gondiiProfile of Thomas E. WellemsPfCRT and the trans-vacuolar proton electrochemical gradient: regulating the access of chloroquine to ferriprotoporphyrin IX.Transporters involved in resistance to antimalarial drugs.PfCRT-mediated drug transport in malarial parasites.Analysis of chloroquine resistance transporter (CRT) isoforms and orthologues in S. cerevisiae yeastPlasmodium falciparum chloroquine resistance transporter is a H+-coupled polyspecific nutrient and drug exporter.Specific inhibition of the plasmodial surface anion channel by dantroleneHeterologous expression of plasmodial proteins for structural studies and functional annotation.Molecular and physiologic basis of quinoline drug resistance in Plasmodium falciparum malariaChloroquine transport in Plasmodium falciparum. 2. Analysis of PfCRT-mediated drug transport using proteoliposomes and a fluorescent chloroquine probe.Drug-resistant malaria: molecular mechanisms and implications for public health.Know your enemy: understanding the role of PfCRT in drug resistance could lead to new antimalarial tactics.In vitro activity of ferroquine is independent of polymorphisms in transport protein genes implicated in quinoline resistance in Plasmodium falciparum.4-N-, 4-S-, and 4-O-chloroquine analogues: influence of side chain length and quinolyl nitrogen pKa on activity vs chloroquine resistant malaria.Chloroquine transport in Plasmodium falciparum. 1. Influx and efflux kinetics for live trophozoite parasites using a novel fluorescent chloroquine probe.A critical role for PfCRT K76T in Plasmodium falciparum verapamil-reversible chloroquine resistance.Verapamil-Sensitive Transport of Quinacrine and Methylene Blue via the Plasmodium falciparum Chloroquine Resistance Transporter Reduces the Parasite's Susceptibility to these Tricyclic Drugs.Absence of association between piperaquine in vitro responses and polymorphisms in the pfcrt, pfmdr1, pfmrp, and pfnhe genes in Plasmodium falciparum.Differences in trans-stimulated chloroquine efflux kinetics are linked to PfCRT in Plasmodium falciparum.Quantitative pH measurements in Plasmodium falciparum-infected erythrocytes using pHluorin.Mutations in transmembrane domains 1, 4 and 9 of the Plasmodium falciparum chloroquine resistance transporter alter susceptibility to chloroquine, quinine and quinidine.Dissecting the components of quinine accumulation in Plasmodium falciparum.
P2860
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P2860
Dictyostelium discoideum expresses a malaria chloroquine resistance mechanism upon transfection with mutant, but not wild-type, Plasmodium falciparum transporter PfCRT.
description
2005 nî lūn-bûn
@nan
2005年の論文
@ja
2005年論文
@yue
2005年論文
@zh-hant
2005年論文
@zh-hk
2005年論文
@zh-mo
2005年論文
@zh-tw
2005年论文
@wuu
2005年论文
@zh
2005年论文
@zh-cn
name
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@ast
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@en
type
label
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@ast
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@en
prefLabel
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@ast
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@en
P2093
P2860
P921
P356
P1476
Dictyostelium discoideum expre ...... falciparum transporter PfCRT.
@en
P2093
Alan R Kimmel
Bronwen Naudé
Joseph A Brzostowski
Thomas E Wellems
P2860
P304
25596-25603
P356
10.1074/JBC.M503227200
P407
P577
2005-05-09T00:00:00Z