Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor
about
Ligand-based virtual screening interface between PyMOL and LiSiCANovel N-allyl/propargyl tetrahydroquinolines: Synthesis via Three-component Cationic Imino Diels-Alder Reaction, Binding Prediction, and Evaluation as Cholinesterase Inhibitors.Development of an in-vivo active reversible butyrylcholinesterase inhibitor.Dual inhibitors of cholinesterases and monoamine oxidases for Alzheimer's disease.Novel Selective Butyrylcholinesterase Inhibitors Incorporating Antioxidant Functionalities as Potential Bimodal Therapeutics for Alzheimer's Disease.Evaluating Fmoc-amino acids as selective inhibitors of butyrylcholinesterase.Comparison of the Binding of Reversible Inhibitors to Human Butyrylcholinesterase and Acetylcholinesterase: A Crystallographic, Kinetic and Calorimetric Study.Proline-Based Carbamates as Cholinesterase Inhibitors.Rapid Mechanistic Evaluation and Parameter Estimation of Putative Inhibitors in a Single-Step Progress-Curve Analysis: The Case of Horse Butyrylcholinesterase.Multiple Ligands Targeting Cholinesterases and β-Amyloid: Synthesis, Biological Evaluation of Heterodimeric Compounds with Benzylamine Pharmacophore.Novel tetrahydroacridine derivatives with iodobenzoic acid moiety as multifunctional acetylcholinesterase inhibitors.Synthesis, pharmacology and molecular docking on multifunctional tacrine-ferulic acid hybrids as cholinesterase inhibitors against Alzheimer's disease.ω-Imidazolyl- and ω-Tetrazolylalkylcarbamates as Inhibitors of Fatty Acid Amide Hydrolase: Biological Activity and in vitro Metabolic Stability.Discovery of (phenylureido)piperidinyl benzamides as prospective inhibitors of bacterial autolysin E from Staphylococcus aureusSynthesis and biological evaluation of 8-hydroxy-2,7-naphthyridin-2-ium salts as novel inhibitors of acetylcholinesterase (AChE) and butyrylcholinesterase (BChE)
P2860
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P2860
Discovery, biological evaluation, and crystal structure of a novel nanomolar selective butyrylcholinesterase inhibitor
description
2014 nî lūn-bûn
@nan
2014 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2014 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2014年の論文
@ja
2014年論文
@yue
2014年論文
@zh-hant
2014年論文
@zh-hk
2014年論文
@zh-mo
2014年論文
@zh-tw
2014年论文
@wuu
name
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@ast
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@en
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@nl
type
label
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@ast
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@en
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@nl
prefLabel
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@ast
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@en
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@nl
P2093
P50
P3181
P356
P1476
Discovery, biological evaluati ...... utyrylcholinesterase inhibitor
@en
P2093
Anja Pišlar
Boris Brus
Jure Stojan
Urban Košak
P304
P3181
P356
10.1021/JM501195E
P407
P577
2014-10-09T00:00:00Z