Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry
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Protein-Templated Fragment Ligations-From Molecular Recognition to Drug Discovery.What is the future for fragment-based drug discovery?Target-directed Dynamic Combinatorial Chemistry: A Study on Potentials and Pitfalls as Exemplified on a Bacterial Target.Redox Control over Acyl Hydrazone Photoswitches.Fragment-Based Drug Design Facilitated by Protein-Templated Click Chemistry: Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin.Insights into the Impact of Linker Flexibility and Fragment Ionization on the Design of CK2 Allosteric Inhibitors: Comparative Molecular Dynamics Simulation Studies.Identification of inhibitors targeting Mycobacterium tuberculosis cell wall biosynthesis via dynamic combinatorial chemistry.Inhibition of the Cysteine Protease Human Cathepsin L by Triazine Nitriles: Amide⋅⋅⋅Heteroarene π-Stacking Interactions and Chalcogen Bonding in the S3 Pocket.Discovery of a Biologically Active Bromodomain Inhibitor by Target-Directed Dynamic Combinatorial Chemistry
P2860
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P2860
Fragment Linking and Optimization of Inhibitors of the Aspartic Protease Endothiapepsin: Fragment-Based Drug Design Facilitated by Dynamic Combinatorial Chemistry
description
2016 nî lūn-bûn
@nan
2016 թուականի Օգոստոսին հրատարակուած գիտական յօդուած
@hyw
2016 թվականի օգոստոսին հրատարակված գիտական հոդված
@hy
2016年の論文
@ja
2016年論文
@yue
2016年論文
@zh-hant
2016年論文
@zh-hk
2016年論文
@zh-mo
2016年論文
@zh-tw
2016年论文
@wuu
name
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@ast
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@en
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@nl
type
label
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@ast
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@en
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@nl
prefLabel
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@ast
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@en
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@nl
P2860
P50
P3181
P356
P1476
Fragment Linking and Optimizat ...... ynamic Combinatorial Chemistry
@en
P2093
Nedyalka Radeva
P2860
P304
P3181
P356
10.1002/ANIE.201603074
P407
P577
2016-08-01T00:00:00Z