The delta-opioid receptor: molecular pharmacology, signal transduction, and the determination of drug efficacy
about
Genetic susceptibility to heroin addiction: a candidate gene association studyRobust optimization of SVM hyperparameters in the classification of bioactive compoundsInhibition of brain [(3)H]cimetidine binding by improgan-like antinociceptive drugs.Ionic storm in hypoxic/ischemic stress: can opioid receptors subside it?Synaptic mechanism for functional synergism between delta- and mu-opioid receptors.Delta-opioid receptor analgesia is independent of microglial activation in a rat model of neuropathic painBiological and conformational evaluation of bifunctional compounds for opioid receptor agonists and neurokinin 1 receptor antagonists possessing two penicillaminesPlasmon resonance studies of agonist/antagonist binding to the human delta-opioid receptor: new structural insights into receptor-ligand interactions.Exploring binding properties of agonists interacting with a δ-opioid receptor.Lipid bilayers on polyacrylamide brushes for inclusion of membrane proteinsδ-Opioid receptors stimulate GLUT1-mediated glucose uptake through Src- and IGF-1 receptor-dependent activation of PI3-kinase signalling in CHO cellsOvarian hormones influence corticotropin releasing factor receptor colocalization with delta opioid receptors in CA1 pyramidal cell dendrites.Design and synthesis of novel hydrazide-linked bifunctional peptides as delta/mu opioid receptor agonists and CCK-1/CCK-2 receptor antagonists.G protein independent phosphorylation and internalization of the delta-opioid receptor.Modulation of gastrointestinal function by MuDelta, a mixed µ opioid receptor agonist/ µ opioid receptor antagonist.Modeling and simulation of the human delta opioid receptor.Design, synthesis, and biological evaluation of novel bifunctional C-terminal-modified peptides for delta/mu opioid receptor agonists and neurokinin-1 receptor antagonists.Imaging of opioid receptors in the central nervous systemKinase cascades and ligand-directed signaling at the kappa opioid receptor.Molecular Pharmacology of δ-Opioid Receptors.The influences of reproductive status and acute stress on the levels of phosphorylated delta opioid receptor immunoreactivity in rat hippocampus.Synthesis of a potent and selective (18)F-labeled delta-opioid receptor antagonist derived from the Dmt-Tic pharmacophore for positron emission tomography imaging.The behavioral effects of a mixed efficacy antinociceptive peptide, VRP26, following chronic administration in mice.The biological activity and metabolic stability of peptidic bifunctional compounds that are opioid receptor agonists and neurokinin-1 receptor antagonists with a cystine moiety.δ-opioid receptor and somatostatin receptor-4 heterodimerization: possible implications in modulation of pain associated signaling.The Opioid System in Temporal Lobe Epilepsy: Functional Role and Therapeutic Potential.Cyclic Opioid Peptides.Exploring the Backbone of Enkephalins To Adjust Their Pharmacological Profile for the δ-Opioid Receptor.Ligands act as pharmacological chaperones and increase the efficiency of delta opioid receptor maturationBioluminescence resonance energy transfer assays reveal ligand-specific conformational changes within preformed signaling complexes containing delta-opioid receptors and heterotrimeric G proteins.Ligand modulation of lateral segregation of a G-protein-coupled receptor into lipid microdomains in sphingomyelin/phosphatidylcholine solid-supported bilayersAn investigation of whether agonist-selective receptor conformations occur with respect to M2 and M4 muscarinic acetylcholine receptor signalling via Gi/o and Gs proteinsIn Vivo Effects of μ Opioid Receptor Agonist/δ Opioid Receptor Antagonist Peptidomimetics Following Acute and Repeated Administration.
P2860
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P2860
The delta-opioid receptor: molecular pharmacology, signal transduction, and the determination of drug efficacy
description
1999 nî lūn-bûn
@nan
1999 թուականի Սեպտեմբերին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի սեպտեմբերին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
The delta-opioid receptor: mol ...... determination of drug efficacy
@ast
The delta-opioid receptor: mol ...... determination of drug efficacy
@en
The delta-opioid receptor: mol ...... determination of drug efficacy
@nl
type
label
The delta-opioid receptor: mol ...... determination of drug efficacy
@ast
The delta-opioid receptor: mol ...... determination of drug efficacy
@en
The delta-opioid receptor: mol ...... determination of drug efficacy
@nl
prefLabel
The delta-opioid receptor: mol ...... determination of drug efficacy
@ast
The delta-opioid receptor: mol ...... determination of drug efficacy
@en
The delta-opioid receptor: mol ...... determination of drug efficacy
@nl
P2093
P1476
The delta-opioid receptor: mol ...... determination of drug efficacy
@en
P2093
F J Ehlert
H I Yamamura
K Hosohata
S M Cowell
T H Burkey
W R Roeske
Y Hosohata
P304
P407
P577
1999-09-01T00:00:00Z