Small molecules showing significant protection of mice against botulinum neurotoxin serotype A
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Metal Ion Modeling Using Classical MechanicsStructural insight into exosite binding and discovery of novel exosite inhibitors of botulinum neurotoxin serotype A through in silico screening.Small-molecule quinolinol inhibitor identified provides protection against BoNT/A in mice.Enhancing the Pharmacokinetic Properties of Botulinum Neurotoxin Serotype A Protease Inhibitors Through Rational DesignDynamin inhibition blocks botulinum neurotoxin type A endocytosis in neurons and delays botulismCargo-delivery platforms for targeted delivery of inhibitor cargos against botulism.Monoclonal Antibodies that Inhibit the Proteolytic Activity of Botulinum Neurotoxin Serotype/B.Substrate-based inhibitors exhibiting excellent protective and therapeutic effects against Botulinum Neurotoxin A intoxicationPaclitaxel is an inhibitor and its boron dipyrromethene derivative is a fluorescent recognition agent for botulinum neurotoxin subtype A.Use of multiple picosecond high-mass molecular dynamics simulations to predict crystallographic B-factors of folded globular proteins.Targeting botulinum A cellular toxicity: a prodrug approach.Targeting bacterial toxins.Current strategies for designing antidotes against botulinum neurotoxins.Challenges in searching for therapeutics against Botulinum Neurotoxins.New Steroidal 4-Aminoquinolines Antagonize Botulinum Neurotoxin Serotype A in Mouse Embryonic Stem Cell Derived Motor Neurons in Post-intoxication Model.Studies on the binding modes of Lassa nucleoprotein complexed with m7GpppG and dTTP by molecular dynamic simulations and free energy calculations.Discovery of a fluorene class of compounds as inhibitors of botulinum neurotoxin serotype E by virtual screening
P2860
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P2860
Small molecules showing significant protection of mice against botulinum neurotoxin serotype A
description
2010 nî lūn-bûn
@nan
2010 թուականի Ապրիլին հրատարակուած գիտական յօդուած
@hyw
2010 թվականի ապրիլին հրատարակված գիտական հոդված
@hy
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
name
Small molecules showing signif ...... otulinum neurotoxin serotype A
@ast
Small molecules showing signif ...... otulinum neurotoxin serotype A
@en
Small molecules showing signif ...... otulinum neurotoxin serotype A
@nl
type
label
Small molecules showing signif ...... otulinum neurotoxin serotype A
@ast
Small molecules showing signif ...... otulinum neurotoxin serotype A
@en
Small molecules showing signif ...... otulinum neurotoxin serotype A
@nl
prefLabel
Small molecules showing signif ...... otulinum neurotoxin serotype A
@ast
Small molecules showing signif ...... otulinum neurotoxin serotype A
@en
Small molecules showing signif ...... otulinum neurotoxin serotype A
@nl
P2093
P2860
P3181
P1433
P1476
Small molecules showing signif ...... otulinum neurotoxin serotype A
@en
P2093
Charles B Millard
James J Schmidt
Jewn Giew Park
Madhusoodana P Nambiar
Shaohua Wang
P2860
P304
P3181
P356
10.1371/JOURNAL.PONE.0010129
P407
P577
2010-04-13T00:00:00Z