Rational design of a peptide agonist that interacts selectively with the orphan receptor, bombesin receptor subtype 3.
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International Union of Pharmacology. LXVIII. Mammalian bombesin receptors: nomenclature, distribution, pharmacology, signaling, and functions in normal and disease statesBombesin-related peptides and their receptors: recent advances in their role in physiology and disease statesInsights into bombesin receptors and ligands: Highlighting recent advancesSystematic optimization of a lead-structure identities for a selective short peptide agonist for the human orphan receptor BRS-3.Bombesin receptor subtype 3 as a potential target for obesity and diabetes.Novel chiral-diazepines function as specific, selective receptor agonists with variable coupling and species variability in human, mouse and rat BRS-3 receptor cells.Pharmacology of putative selective hBRS-3 receptor agonists for human bombesin receptors (BnR): affinities, potencies and selectivity in multiple native and BnR transfected cells.mRNA display selection and solid-phase synthesis of Fc-binding cyclic peptide affinity ligands.Bombesin receptor subtype-3 agonists stimulate the growth of lung cancer cells and increase EGF receptor tyrosine phosphorylation.Pharmacology and selectivity of various natural and synthetic bombesin related peptide agonists for human and rat bombesin receptors differs.The molecular basis for high affinity of a universal ligand for human bombesin receptor (BnR) family members.GRPR-targeted Protein Contrast Agents for Molecular Imaging of Receptor Expression in Cancers by MRIMolecular basis for agonist selectivity and activation of the orphan bombesin receptor subtype 3 receptor.Bombesin inhibits alveolarization and promotes pulmonary fibrosis in newborn mice.Characterization of putative GRP- and NMB-receptor antagonist's interaction with human receptors.A selective human bombesin receptor subtype-3 peptide agonist mediates CREB phosphorylation and transactivation.Molecular basis for high affinity and selectivity of peptide antagonist, Bantag-1, for the orphan BB3 receptor.Gastrin-releasing peptide is a modulatory neurotransmitter of the descending phase of the peristaltic reflex.
P2860
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P2860
Rational design of a peptide agonist that interacts selectively with the orphan receptor, bombesin receptor subtype 3.
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2000 nî lūn-bûn
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2000 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
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2000 թվականի դեկտեմբերին հրատարակված գիտական հոդված
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2000年の論文
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name
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@ast
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@en
type
label
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@ast
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@en
prefLabel
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@ast
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@en
P2093
P2860
P356
P1476
Rational design of a peptide a ...... , bombesin receptor subtype 3.
@en
P2093
Igarashi H
Pradhan TK
P2860
P304
P356
10.1074/JBC.M008737200
P407
P577
2000-12-08T00:00:00Z