about
Transport proteins determine drug sensitivity and resistance in a protozoan parasite, Trypanosoma bruceiInteraction of monobenzamidine-linked trypanocides with the Trypanosoma brucei P2 aminopurine transporterResistance to pentamidine in Leishmania mexicana involves exclusion of the drug from the mitochondrion.Nucleoside and nucleobase transporters in parasitic protozoa.Purine and pyrimidine transport in pathogenic protozoa: from biology to therapy.Aromatic diamidines as antiparasitic agents.Functional expression of TcoAT1 reveals it to be a P1-type nucleoside transporter with no capacity for diminazene uptakeTransporters for drug delivery and as drug targets in parasitic protozoa.Trypanosoma brucei aquaglyceroporin 2 is a high-affinity transporter for pentamidine and melaminophenyl arsenic drugs and the main genetic determinant of resistance to these drugs.Neglected disease - african sleeping sickness: recent synthetic and modeling advances.Functional analysis of drug resistance-associated mutations in the Trypanosoma brucei adenosine transporter 1 (TbAT1) and the proposal of a structural model for the protein.9-(2'-Deoxy-2'-Fluoro-β-d-Arabinofuranosyl) Adenine Is a Potent Antitrypanosomal Adenosine Analogue That Circumvents Transport-Related Drug Resistance.T-2307, a novel arylamidine, is transported into Candida albicans by a high-affinity spermine and spermidine carrier regulated by Agp2.Uptake of T-2307, a novel arylamidine, in Candida albicans.Functional expression and characterization of a purine nucleobase transporter gene from Leishmania major.
P2860
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P2860
description
1999 nî lūn-bûn
@nan
1999 թուականի Դեկտեմբերին հրատարակուած գիտական յօդուած
@hyw
1999 թվականի դեկտեմբերին հրատարակված գիտական հոդված
@hy
1999年の論文
@ja
1999年論文
@yue
1999年論文
@zh-hant
1999年論文
@zh-hk
1999年論文
@zh-mo
1999年論文
@zh-tw
1999年论文
@wuu
name
A drug resistance determinant in Trypanosoma brucei.
@ast
A drug resistance determinant in Trypanosoma brucei.
@en
type
label
A drug resistance determinant in Trypanosoma brucei.
@ast
A drug resistance determinant in Trypanosoma brucei.
@en
prefLabel
A drug resistance determinant in Trypanosoma brucei.
@ast
A drug resistance determinant in Trypanosoma brucei.
@en
P1476
A drug resistance determinant in Trypanosoma brucei
@en
P2093
N S Carter
P304
P356
10.1016/S0966-842X(99)01643-1
P577
1999-12-01T00:00:00Z