Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H₄ and the ion channel serotonin 5-HT₃A.
about
Diazepam-bound GABAA receptor models identify new benzodiazepine binding-site ligandsCrystal structure-based virtual screening for fragment-like ligands of the human histamine H(1) receptorA Role for Fragment-Based Drug Design in Developing Novel Lead Compounds for Central Nervous System TargetsDiscovery of β2 Adrenergic Receptor Ligands Using Biosensor Fragment Screening of Tagged Wild-Type Receptor.Fragment-based lead discovery on G-protein-coupled receptors.Histamine H4 receptor ligands and their potential therapeutic applications: an update.Structure-based and fragment-based GPCR drug discovery.Histamine H4 receptor ligands: future applications and state of art.Combination histamine and serotonin treatment after simulated childbirth injury improves stress urinary incontinence.Design, synthesis, and structure-activity relationships of highly potent 5-HT₃ receptor ligands.Exploring G Protein-Coupled Receptors (GPCRs) Ligand Space via Cheminformatics Approaches: Impact on Rational Drug Design.Structure-based virtual screening for fragment-like ligands of the G protein-coupled histamine H4 receptor
P2860
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P2860
Fragment library screening reveals remarkable similarities between the G protein-coupled receptor histamine H₄ and the ion channel serotonin 5-HT₃A.
description
2011 nî lūn-bûn
@nan
2011 թուականի Յուլիսին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի հուլիսին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@ast
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@en
type
label
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@ast
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@en
prefLabel
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@ast
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@en
P2093
P2860
P1476
Fragment library screening rev ...... ion channel serotonin 5-HT₃A.
@en
P2093
Andrew J Thompson
Gerdien E de Kloe
Henry F Vischer
Iwan J P de Esch
Jacqueline E van Muijlwijk-Koezen
Linda Silvestri
Mark H P Verheij
Obbe P Zuiderveld
Rogier A Smits
P2860
P304
P356
10.1016/J.BMCL.2011.06.123
P407
P577
2011-07-02T00:00:00Z