Structure-activity relationship study of 2,4-diaminothiazoles as Cdk5/p25 kinase inhibitors.

Structure-activity relationship study of 2,4-diaminothiazoles as Cdk5/p25 kinase inhibitors.

Item
http://www.wikidata.org/entity/Q34706737
Development of Highly Potent and Selective Diaminothiazole Inhibitors of Cyclin-Dependent KinasesDiscovery of thienoquinolone derivatives as selective and ATP non-competitive CDK5/p25 inhibitors by structure-based virtual screeningFrom on-target to off-target activity: identification and optimisation of Trypanosoma brucei GSK3 inhibitors and their characterisation as anti-Trypanosoma brucei drug discovery lead molecules.Diaminothiazoles modify Tau phosphorylation and improve the tauopathy in mouse modelsApproaches to efficiently estimate solvation and explicit water energetics in ligand binding: the use of WaterMap.Drug discovery and human African trypanosomiasis: a disease less neglected?Determination of kinetic parameters and structure-activity relationships of ginsenosides as inhibitors of cyclin-dependent kinase 5/p25 using ultra-pressure liquid chromatography with triple quadrupole tandem mass spectrometry.Consensus models for CDK5 inhibitors in silico and their application to inhibitor discovery.Several human cyclin-dependent kinase inhibitors, structurally related to roscovitine, are new anti-malarial agents.
P2860

Structure-activity relationship study of 2,4-diaminothiazoles as Cdk5/p25 kinase inhibitors.

Item
http://www.wikidata.org/entity/Q34706737
description
2011 nî lūn-bûn
@nan
2011 թուականի Փետրուարին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի փետրվարին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@ast
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@en
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@nl
type
label
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@ast
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@en
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@nl
prefLabel
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@ast
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@en
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@nl
P1433
P1476
P2093
P2860
P304
P31
P356
P407
P433
P478
P577
P5875
P698
P932
P356
P1433
P1476
Structure-activity relationshi ...... as Cdk5/p25 kinase inhibitors.
@en
P2093
P2860
P304
P31
P356
10.1016/J.BMCL.2011.01.140
P407
P433
P478
P577
P5875
P698
P932