Investigation of unanticipated alkylation at the N(π) position of a histidyl residue under Mitsunobu conditions and synthesis of orthogonally protected histidine analogues.
about
Neighbor-directed histidine N (τ)-alkylation: A route to imidazolium-containing phosphopeptide macrocyclesDe novo design and synthesis of ultra-short peptidomimetic antibiotics having dual antimicrobial and anti-inflammatory activities.Mitsunobu mischief: neighbor-directed histidine N(τ)-alkylation provides access to peptides containing selectively functionalized imidazolium heterocycles.Effects on polo-like kinase 1 polo-box domain binding affinities of peptides incurred by structural variation at the phosphoamino acid position.Design of new acid-activated cell-penetrating peptides for tumor drug deliveryMono-anionic phosphopeptides produced by unexpected histidine alkylation exhibit high Plk1 polo-box domain-binding affinities and enhanced antiproliferative effects in HeLa cells.Peptide-based inhibitors of Plk1 polo-box domain containing mono-anionic phosphothreonine esters and their pivaloyloxymethyl prodrugs.Phosphatase-Stable Phosphoamino Acid Mimetics That Enhance Binding Affinities with the Polo-Box Domain of Polo-like Kinase 1.Application of oxime-diversification to optimize ligand interactions within a cryptic pocket of the polo-like kinase 1 polo-box domain.Enhancing polo-like kinase 1 selectivity of polo-box domain-binding peptides.Design and Synthesis of Fmoc-Thr[PO(OH)(OPOM)] for the Preparation of Peptide Prodrugs Containing Phosphothreonine in Fully Protected Form
P2860
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P2860
Investigation of unanticipated alkylation at the N(π) position of a histidyl residue under Mitsunobu conditions and synthesis of orthogonally protected histidine analogues.
description
2011 nî lūn-bûn
@nan
2011 թուականի Հոկտեմբերին հրատարակուած գիտական յօդուած
@hyw
2011 թվականի հոտեմբերին հրատարակված գիտական հոդված
@hy
2011年の論文
@ja
2011年論文
@yue
2011年論文
@zh-hant
2011年論文
@zh-hk
2011年論文
@zh-mo
2011年論文
@zh-tw
2011年论文
@wuu
name
Investigation of unanticipated ...... protected histidine analogues.
@ast
Investigation of unanticipated ...... protected histidine analogues.
@en
type
label
Investigation of unanticipated ...... protected histidine analogues.
@ast
Investigation of unanticipated ...... protected histidine analogues.
@en
prefLabel
Investigation of unanticipated ...... protected histidine analogues.
@ast
Investigation of unanticipated ...... protected histidine analogues.
@en
P2860
P356
P1476
Investigation of unanticipated ...... protected histidine analogues.
@en
P2093
Terrence R Burke
P2860
P304
P356
10.1021/JO201599C
P407
P50
P577
2011-10-03T00:00:00Z