Structure-activity relationships of truncated adenosine derivatives as highly potent and selective human A3 adenosine receptor antagonists.
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Recent developments in adenosine receptor ligands and their potential as novel drugsActivation of adenosine low-affinity A3 receptors inhibits the enteric short interplexus neural circuit triggered by histamine.Functionalized congeners of A3 adenosine receptor-selective nucleosides containing a bicyclo[3.1.0]hexane ring system.Truncated (N)-Methanocarba Nucleosides as A(1) Adenosine Receptor Agonists and Partial Agonists: Overcoming Lack of a Recognition ElementSynthesis and anti-renal fibrosis activity of conformationally locked truncated 2-hexynyl-N(6)-substituted-(N)-methanocarba-nucleosides as A3 adenosine receptor antagonists and partial agonists.The A3 adenosine receptor as multifaceted therapeutic target: pharmacology, medicinal chemistry, and in silico approaches.Discovery of Molecular Therapeutics for Glaucoma: Challenges, Successes, and Promising Directions.
P2860
Q27687253-56220C97-5126-4F6B-9BE2-6BAC158E8BE8Q33771708-21018874-12CC-46BF-9FD8-CF6FA349FA53Q35029175-A5C62755-3115-4B63-8D40-C8C9268A0612Q35165684-96D49710-F29F-4F6B-8BD9-F75485D8504AQ37637798-98C0A3D4-33D8-4519-8D87-4ACF4AF47968Q37957791-7B15E9AE-4434-4D73-9716-25DC4C65ADB3Q38584194-DDDCC38D-FBA1-4494-9BC2-4BDA00DD8CC7
P2860
Structure-activity relationships of truncated adenosine derivatives as highly potent and selective human A3 adenosine receptor antagonists.
description
2009 nî lūn-bûn
@nan
2009年の論文
@ja
2009年論文
@yue
2009年論文
@zh-hant
2009年論文
@zh-hk
2009年論文
@zh-mo
2009年論文
@zh-tw
2009年论文
@wuu
2009年论文
@zh
2009年论文
@zh-cn
name
Structure-activity relationshi ...... denosine receptor antagonists.
@ast
Structure-activity relationshi ...... denosine receptor antagonists.
@en
type
label
Structure-activity relationshi ...... denosine receptor antagonists.
@ast
Structure-activity relationshi ...... denosine receptor antagonists.
@en
prefLabel
Structure-activity relationshi ...... denosine receptor antagonists.
@ast
Structure-activity relationshi ...... denosine receptor antagonists.
@en
P2093
P2860
P1476
Structure-activity relationshi ...... denosine receptor antagonists.
@en
P2093
Cara L Heller
Hea Ok Kim
Kenneth A Jacobson
Lak Shin Jeong
Moshe Chinn
Sang Kook Lee
Seung Ah Choe
Shantanu Pal
Won Jun Choi
P2860
P304
P356
10.1016/J.BMC.2009.03.034
P407
P577
2009-03-25T00:00:00Z