Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity. - Wikidata - awgldk - TriplyDB

Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity.

Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity.

http://www.wikidata.org/entity/Q37366806

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Recent developments in drug discovery for leishmaniasis and human African trypanosomiasis Structural aspects of intermolecular interactions in the solid state of 1,4-dibenzylpiperazines bearing nitrile or amidine groups Analogs of pentamidine as potential anti-Pneumocystis chemotherapeutics.3,1-Benzothiazines, 1,4-Benzodioxines and 1,4-Benzoxazines as Inhibitors of Matriptase-2: Outcome of a Focused Screening Approach.Pentamidine analogs as inhibitors of [(3)H]MK-801 and [(3)H]ifenprodil binding to rat brain NMDA receptors.Diamidines versus Monoamidines as Anti-Pneumocystis Agents: An in Vivo Study.From multiply active natural product to candidate drug? Antibacterial (and other) minor groove binders for DNA.Activity of diimidazoline amides against African trypanosomiasis.Alkanediamide-Linked Bisbenzamidines Are Promising Antiparasitic Agents.Potential of bisbenzimidazole-analogs toward metronidazole-resistant Trichomonas vaginalis isolates.A Short Peptide Inhibitor as an Activity-Based Probe for Matriptase-2.

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Synthesis and SAR of alkanediamide-linked bisbenzamidines with anti-trypanosomal and anti-pneumocystis activity.

http://www.wikidata.org/entity/Q37366806

description

article científic

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article scientifique

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articolo scientifico

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artigo científico

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bilimsel makale

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scientific article published on 23 August 2009

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vedecký článok

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vetenskaplig artikel

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videnskabelig artikel

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vědecký článek

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name

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

@en

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

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type

label

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

@en

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

@nl

prefLabel

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

@en

Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

@nl

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J.BMCL.2009.08.073

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Bioorganic & Medicinal Chemistry Letters

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Synthesis and SAR of alkanedia ...... nd anti-pneumocystis activity.

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Cyrus J Bacchi

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Donna Rattendi

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Indira Londono

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Jean Jacques Vanden Eynde

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Lakshman Mazumder

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Margaret S Collins

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Nigel Yarlett

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Tien L Huang

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Effects of analogs of the DNA minor groove binder Hoechst 33258 on topoisomerase II and I mediated activities.

Highly active anti-Pneumocystis carinii compounds in a library of novel piperazine-linked bisbenzamidines and related compounds.

Anti-plasmodial and anti-leishmanial activity of conformationally restricted pentamidine congeners.

Novel bisbenzimidazoles with antileishmanial effectiveness.

In vitro selection and in vivo efficacy of piperazine- and alkanediamide-linked bisbenzamidines against Pneumocystis pneumonia in mice.

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scholarly article

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10.1016/J.BMCL.2009.08.073

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Melanie T. Cushion

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2009-08-23T00:00:00Z

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