Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
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Exploration of Novel Inhibitors for Class I Histone Deacetylase Isoforms by QSAR Modeling and Molecular Dynamics Simulation AssaysSynthesis and biological evaluation of largazole analogues with modified surface recognition cap groupsComparative pharmacokinetic properties and antitumor activity of the marine HDACi Largazole and Largazole peptide isostereVariable active site loop conformations accommodate the binding of macrocyclic largazole analogues to HDAC8Modular synthesis and biological activity of pyridyl-based analogs of the potent Class I Histone Deacetylase Inhibitor Largazole.Synthesis and biological evaluation of largazole zinc-binding group analogs.Natural and Synthetic Macrocyclic Inhibitors of the Histone Deacetylase Enzymes.Largazole Analogues as Histone Deacetylase Inhibitors and Anticancer Agents: An Overview of Structure-Activity Relationships.
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Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
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article científic
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article scientifique
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articolo scientifico
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artigo científico
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bilimsel makale
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scientific article published on 18 June 2013
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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name
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@en
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@nl
type
label
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@en
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@nl
prefLabel
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@en
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@nl
P2093
P2860
P1476
Synthesis and HDAC inhibitory activity of isosteric thiazoline-oxazole largazole analogs.
@en
P2093
Albert A Bowers
Guillermina Estiu
James E Bradner
Jennifer M Guerra-Bubb
Olaf Wiest
Robert M Williams
Ronald Paranal
William B Smith
P2860
P304
P356
10.1016/J.BMCL.2013.06.012
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P577
2013-06-18T00:00:00Z