Inhibition of heterotrimeric G protein signaling by a small molecule acting on Galpha subunit.
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Calcium-sensing receptors signal constitutive macropinocytosis and facilitate the uptake of NOD2 ligands in macrophages.The oligomeric state sets GABA(B) receptor signalling efficacyLigand-based peptide design and combinatorial peptide libraries to target G protein-coupled receptorsInhibitory G proteins and their receptors: emerging therapeutic targets for obesity and diabetes.A critical role of Gbetagamma in tumorigenesis and metastasis of breast cancer.Atypical signaling and functional desensitization response of MAS receptor to peptide ligands.Functional interaction between angiotensin II receptor type 1 and chemokine (C-C motif) receptor 2 with implications for chronic kidney diseaseAssessing Gonadotropin Receptor Function by Resonance Energy Transfer-Based Assays.Heteromeric MT1/MT2 melatonin receptors modulate photoreceptor function.Interaction of Protease-Activated Receptor 2 with G Proteins and β-Arrestin 1 Studied by Bioluminescence Resonance Energy Transfer.Probing heterotrimeric G protein activation: applications to biased ligands.BRET biosensors to study GPCR biology, pharmacology, and signal transduction.Molecular targeting of Gα and Gβγ subunits: a potential approach for cancer therapeutics.Biophysical Detection of Diversity and Bias in GPCR Function.Genetic, structural, and molecular insights into the function of ras of complex proteins domains.A cell-permeable inhibitor to trap Gαq proteins in the empty pocket conformation.Crosstalk between angiotensin and the nonamyloidogenic pathway of Alzheimer's amyloid precursor protein.The Gαi-GIV binding interface is a druggable protein-protein interactionLysophosphatidic acid increases proximal tubule cell secretion of profibrotic cytokines PDGF-B and CTGF through LPA2- and Gαq-mediated Rho and αvβ6 integrin-dependent activation of TGF-βReceptor-G protein interaction studied by bioluminescence resonance energy transfer: lessons from protease-activated receptor 1.The vasoactive peptides urotensin II and urotensin II-related peptide regulate astrocyte activity through common and distinct mechanisms: involvement in cell proliferation.Potent and Selective Peptide-based Inhibition of the G Protein Gαq.Molecular Approaches To Target GPCRs in Cancer Therapy.Bruton's tyrosine kinase and RAC1 promote cell survival in MLL-rearranged acute myeloid leukemia.
P2860
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P2860
Inhibition of heterotrimeric G protein signaling by a small molecule acting on Galpha subunit.
description
article científic
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article scientifique
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articolo scientifico
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artigo científico
@pt
bilimsel makale
@tr
scientific article published on 31 July 2009
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vedecký článok
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vetenskaplig artikel
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videnskabelig artikel
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vědecký článek
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name
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@en
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@nl
type
label
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@en
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@nl
prefLabel
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@en
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@nl
P2093
P2860
P356
P1476
Inhibition of heterotrimeric G ...... cule acting on Galpha subunit.
@en
P2093
Christian Gespach
Eric Ferrandis
Grégoire Pierre Prévost
Jean-Louis Banères
Jean-Philippe Pin
Marjorie Damian
Mohammed Akli Ayoub
Olivier De Wever
Olivier Lavergne
P2860
P304
29136-29145
P356
10.1074/JBC.M109.042333
P407
P577
2009-07-31T00:00:00Z