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σ-1 receptor at the mitochondrial-associated endoplasmic reticulum membrane is responsible for mitochondrial metabolic regulationSigma1 receptor antagonists determine the behavioral pattern of the methamphetamine-induced stereotypy in miceAntagonist action of progesterone at σ-receptors in the modulation of voltage-gated sodium channelsPurification, molecular cloning, and expression of the mammalian sigma1-binding siteAn unambiguous assay for the cloned human sigma1 receptor reveals high affinity interactions with dopamine D4 receptor selective compounds and a distinct structure-affinity relationship for butyrophenonesSigma receptor agonists provide neuroprotection in vitro by preserving bcl-2Role of sigma-1 receptor C-terminal segment in inositol 1,4,5-trisphosphate receptor activation: constitutive enhancement of calcium signaling in MCF-7 tumor cellsThe sigma-receptor antagonist BD-1063 decreases ethanol intake and reinforcement in animal models of excessive drinkingThe dextromethorphan analog dimemorfan attenuates kainate-induced seizures via sigma1 receptor activation: comparison with the effects of dextromethorphanAntitussive activity of sigma-1 receptor agonists in the guinea-pigDifferentiation of sigma ligand-activated receptor subtypes that modulate NMDA-evoked [3H]-noradrenaline release in rat hippocampal slicesNo association between the sigma receptor type 1 gene and schizophrenia: results of analysis and meta-analysis of case-control studiesDifferential involvement of the sigma(1) (sigma(1)) receptor in the anti-amnesic effect of neuroactive steroids, as demonstrated using an in vivo antisense strategy in the mouseSiramesine triggers cell death through destabilisation of mitochondria, but not lysosomesThe sigma-1 receptor is enriched in postsynaptic sites of C-terminals in mouse motoneurons. An anatomical and behavioral study4-aroylpiperidines and 4-(α-hydroxyphenyl)piperidines as selective sigma-1 receptor ligands: synthesis, preliminary pharmacological evaluation and computational studiesActivation of the Sigma-1 receptor by haloperidol metabolites facilitates brain-derived neurotrophic factor secretion from human astrogliaThe novel ketamine analog methoxetamine produces dissociative-like behavioral effects in rodents.Bi-phasic intensity-dependent opioid-mediated neural amplitude changes in the chinchilla cochlea: partial blockade by an N-Methyl-D-Aspartate (NMDA)-receptor antagonistσ1 receptor ligands control a switch between passive and active threat responses.Effects of (+)-pentazocine and 1,3-di-o-tolylguanidine (DTG), sigma (sigma) ligands, on micturition in anaesthetized rats.Development of molecular probes for imaging sigma-2 receptors in vitro and in vivo.Cyclic adenosine monophosphate response element-binding protein phosphorylation and neuroprotection by 4-phenyl-1-(4-phenylbutyl) piperidine (PPBP).The σ2 receptor: a novel protein for the imaging and treatment of cancer.Synthesis and receptor profiling of Stemona alkaloid analogues reveal a potent class of sigma ligandsAnimal models of focal dystonia.Targeted pancreatic cancer therapy with the small molecule drug conjugate SW IV-134.Identification of the gene that codes for the σ2 receptor.Current hypotheses on sigma receptors and their physiological role: possible implications in psychiatry.Radiosynthesis and biological evaluation of a promising sigma(2)-receptor ligand radiolabeled with fluorine-18 or iodine-125 as a PET/SPECT probe for imaging breast cancer.Neurosteroids, via sigma receptors, modulate the [3H]norepinephrine release evoked by N-methyl-D-aspartate in the rat hippocampus.SA 4503 attenuates cocaine-induced hyperactivity and enhances methamphetamine substitution for a cocaine discriminative stimulusTargeting ligand-operated chaperone sigma-1 receptors in the treatment of neuropsychiatric disorders.Activation of σ-receptors induces binge-like drinking in Sardinian alcohol-preferring ratsThe sigma receptor agonist SA4503 both attenuates and enhances the effects of methamphetamine.The novel sigma-2 receptor ligand SW43 stabilizes pancreas cancer progression in combination with gemcitabine.A Role for Sigma Receptors in Stimulant Self Administration and Addiction.Intrathecal treatment with sigma1 receptor antagonists reduces formalin-induced phosphorylation of NMDA receptor subunit 1 and the second phase of formalin test in miceCharacterization and evaluation of two novel fluorescent sigma-2 receptor ligands as proliferation probes.Central neuropeptide Y and the sigma ligand, JO 1784, reverse corticotropin-releasing factor-induced inhibition of gastric acid secretion in rats.
P2860
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P2860
description
article científic
@ca
article scientifique
@fr
articolo scientifico
@it
artigo científico
@pt
bilimsel makale
@tr
scientific article published on December 1990
@en
vedecký článok
@sk
vetenskaplig artikel
@sv
videnskabelig artikel
@da
vědecký článek
@cs
name
Sigma receptors: biology and function.
@en
Sigma receptors: biology and function.
@nl
type
label
Sigma receptors: biology and function.
@en
Sigma receptors: biology and function.
@nl
prefLabel
Sigma receptors: biology and function.
@en
Sigma receptors: biology and function.
@nl
P2093
P1476
Sigma receptors: biology and function.
@en
P2093
P304
P577
1990-12-01T00:00:00Z