Substrate inhibition kinetics in drug metabolism reactions.
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Regioselective Glucuronidation of Diosmetin and Chrysoeriol by the Interplay of Glucuronidation and Transport in UGT1A9-Overexpressing HeLa CellsIn Silico Prediction of Human Sulfotransferase 1E1 Activity Guided by Pharmacophores from Molecular Dynamics Simulations.Substrate selectivity of drug-metabolizing cytochrome P450s predicted from crystal structures and in silico modeling.Crystal structures of human sulfotransferases: insights into the mechanisms of action and substrate selectivity.Reaction phenotyping to assess victim drug-drug interaction risks.In vitro-in silico-based analysis of the dose-dependent in vivo oestrogenicity of the soy phytoestrogen genistein in humans.Regioselective glucuronidation of gingerols by human liver microsomes and expressed UDP-glucuronosyltransferase enzymes: reaction kinetics and activity correlation analyses for UGT1A9 and UGT2B7.Glucuronidation of capsaicin by liver microsomes and expressed UGT enzymes: reaction kinetics, contribution of individual enzymes and marked species differences.Chemical inhibition and stable knock-down of efflux transporters leads to reduced glucuronidation of wushanicaritin in UGT1A1-overexpressing HeLa cells: the role of breast cancer resistance protein (BCRP) and multidrug resistance-associated proteinsLow Potential of Basimglurant to Be Involved in Drug-Drug Interactions: Influence of Non-Michaelis-Menten P450 Kinetics on Fraction Metabolized.Glucuronidation of macelignan by human liver microsomes and expressed UGT enzymes: identification of UGT1A1 and 2B7 as the main contributing enzymes.
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Substrate inhibition kinetics in drug metabolism reactions.
description
article científic
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article scientifique
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articol științific
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articolo scientifico
@it
artigo científico
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artigo científico
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artigo científico
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artikel ilmiah
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artikull shkencor
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artículo científico
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name
Substrate inhibition kinetics in drug metabolism reactions.
@en
Substrate inhibition kinetics in drug metabolism reactions.
@nl
type
label
Substrate inhibition kinetics in drug metabolism reactions.
@en
Substrate inhibition kinetics in drug metabolism reactions.
@nl
prefLabel
Substrate inhibition kinetics in drug metabolism reactions.
@en
Substrate inhibition kinetics in drug metabolism reactions.
@nl
P2860
P1476
Substrate inhibition kinetics in drug metabolism reactions.
@en
P2093
Baojian Wu
P2860
P304
P356
10.3109/03602532.2011.615320
P407
P577
2011-09-30T00:00:00Z