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RVX-208, an inducer of ApoA-I in humans, is a BET bromodomain antagonistStructure of human Sp140 PHD finger: an atypical fold interacting with Pin1SET1 and p300 act synergistically, through coupled histone modifications, in transcriptional activation by p53Epimutational profile of hematologic malignancies as attractive target for new epigenetic therapiesOpen access chemical probes for epigenetic targetsBromodomain proteins in HIV infectionCombating the epigenome: epigenetic drugs against non-Hodgkin's lymphomaThe bromodomain: from epigenome reader to druggable targetMechanisms of Histone Deacetylase Inhibitor-Regulated Gene Expression in Cancer CellsEpigenetic mechanisms in mood disorders: targeting neuroplasticityOptimization of 3,5-Dimethylisoxazole Derivatives as Potent Bromodomain LigandsCyclin-Dependent Kinase Inhibitor Dinaciclib Interacts with the Acetyl-Lysine Recognition Site of BromodomainsDiscovery of Novel Small-Molecule Inhibitors of BRD4 Using Structure-Based Virtual ScreeningBinding of the histone chaperone ASF1 to the CBP bromodomain promotes histone acetylationObserved bromodomain flexibility reveals histone peptide- and small molecule ligand-compatible forms of ATAD2Discovery and Optimization of a Selective Ligand for the Switch/Sucrose Nonfermenting-Related Bromodomains of Polybromo Protein-1 by the Use of Virtual Screening and Hydration AnalysisAcetylation Reader Proteins: Linking Acetylation Signaling to Genome Maintenance and CancerNovel therapeutic strategies for multiple myelomaThe mechanisms behind the therapeutic activity of BET bromodomain inhibitionDiscovery and optimization of small-molecule ligands for the CBP/p300 bromodomainsTowards an understanding of the structure and function of MTA1Inhibition of BET bromodomains as a therapeutic strategy for cancer drug discoveryOpen access target validation is a more efficient way to accelerate drug discoverySPOTing Acetyl-Lysine Dependent InteractionsSensitivity and engineered resistance of myeloid leukemia cells to BRD9 inhibitionThe C-terminal domain of Brd2 is important for chromatin interaction and regulation of transcription and alternative splicing.Binding hotspots of BAZ2B bromodomain: Histone interaction revealed by solution NMR driven docking.Cocaine Administration and Its Withdrawal Enhance the Expression of Genes Encoding Histone-Modifying Enzymes and Histone Acetylation in the Rat Prefrontal Cortex.In silico analysis of protein Lys-N(𝜀)-acetylation in plants.Accelerated chromatin biochemistry using DNA-barcoded nucleosome libraries.Transcriptional/epigenetic regulator CBP/p300 in tumorigenesis: structural and functional versatility in target recognition.Modification of enhancer chromatin: what, how, and why?Epigenomics of macrophages.BET bromodomain inhibitors: a patent review.The bromodomain of Gcn5 regulates site specificity of lysine acetylation on histone H3Selective Small Molecule Induced Degradation of the BET Bromodomain Protein BRD4.New roles for old modifications: emerging roles of N-terminal post-translational modifications in development and disease.Brd4 is essential for IL-1β-induced inflammation in human airway epithelial cellsHistones: at the crossroads of peptide and protein chemistry.Polycomb-mediated silencing in neuroendocrine prostate cancer.
P2860
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P2860
description
article científic
@ca
article scientifique
@fr
articol științific
@ro
articolo scientifico
@it
artigo científico
@gl
artigo científico
@pt
artigo científico
@pt-br
artikel ilmiah
@id
artikull shkencor
@sq
artículo científico
@es
name
The bromodomain interaction module.
@en
type
label
The bromodomain interaction module.
@en
prefLabel
The bromodomain interaction module.
@en
P2860
P1433
P1476
The bromodomain interaction module.
@en
P2860
P304
P356
10.1016/J.FEBSLET.2012.04.045
P407
P577
2012-05-03T00:00:00Z