What is biased efficacy? Defining the relationship between intrinsic efficacy and free energy coupling.
about
Functional competence of a partially engaged GPCR-β-arrestin complexPharmacological Profile of Nociceptin/Orphanin FQ Receptors Interacting with G-Proteins and β-Arrestins 2.The novel PAR2 ligand C391 blocks multiple PAR2 signalling pathways in vitro and in vivo.G Protein-coupled Receptor Biased Agonism.The β-Arrestins: Multifunctional Regulators of G Protein-coupled ReceptorsThermodynamics of GPCR activation.Molecular Pharmacology of δ-Opioid Receptors.Allosteric nanobodies reveal the dynamic range and diverse mechanisms of G-protein-coupled receptor activationA Practical Guide to Approaching Biased Agonism at G Protein Coupled Receptors.Systematic errors in detecting biased agonism: Analysis of current methods and development of a new model-free approach.Biased signalling: from simple switches to allosteric microprocessors.Modelling and simulation of biased agonism dynamics at a G protein-coupled receptor.An evaluation of the operational model when applied to quantify functional selectivity.Evaluation of affinity interaction between small molecules and platelets by open tubular affinity capillary electrochromatography.
P2860
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P2860
What is biased efficacy? Defining the relationship between intrinsic efficacy and free energy coupling.
description
2014 nî lūn-bûn
@nan
2014年の論文
@ja
2014年学术文章
@wuu
2014年学术文章
@zh-cn
2014年学术文章
@zh-hans
2014年学术文章
@zh-my
2014年学术文章
@zh-sg
2014年學術文章
@yue
2014年學術文章
@zh
2014年學術文章
@zh-hant
name
What is biased efficacy? Defin ...... cacy and free energy coupling.
@en
type
label
What is biased efficacy? Defin ...... cacy and free energy coupling.
@en
prefLabel
What is biased efficacy? Defin ...... cacy and free energy coupling.
@en
P50
P1476
What is biased efficacy? Defin ...... icacy and free energy coupling
@en
P2093
H Ongun Onaran
P304
P356
10.1016/J.TIPS.2014.09.010
P577
2014-10-30T00:00:00Z