Synthesis and biological activity of optically active NCL-1, a lysine-specific demethylase 1 selective inhibitor.

Synthesis and biological activity of optically active NCL-1, a lysine-specific demethylase 1 selective inhibitor.

Item
http://www.wikidata.org/entity/Q39608783
Small-molecular modulators of cancer-associated epigenetic mechanisms.Lysine-specific demethylase 1-selective inactivators: protein-targeted drug delivery mechanism.An overview of phenylcyclopropylamine derivatives: biochemical and biological significance and recent developments.Small molecule epigenetic inhibitors targeted to histone lysine methyltransferases and demethylases.Epigenetic pathway targets for the treatment of disease: accelerating progress in the development of pharmacological tools: IUPHAR Review 11.Novel KDM1A inhibitors induce differentiation and apoptosis of glioma stem cells via unfolded protein response pathway.Epigenetics: A primer for clinicians.TCPs: privileged scaffolds for identifying potent LSD1 inhibitors for cancer therapy.Synthesis, LSD1 Inhibitory Activity, and LSD1 Binding Model of Optically Pure Lysine-PCPA Conjugates.Structure-activity study for (bis)ureidopropyl- and (bis)thioureidopropyldiamine LSD1 inhibitors with 3-5-3 and 3-6-3 carbon backbone architecturesThe KDM1A histone demethylase is a promising new target for the epigenetic therapy of medulloblastoma.Histone Lysine Demethylase Inhibitors.Structural insight into inhibitors of flavin adenine dinucleotide-dependent lysine demethylases.Low molecular weight amidoximes that act as potent inhibitors of lysine-specific demethylase 1Targeting histone methyltransferase and demethylase in acute myeloid leukemia therapy.C-H activation enables a rapid structure-activity relationship study of arylcyclopropyl amines for potent and selective LSD1 inhibitors.Regulation of tissue factor pathway inhibitor-2 (TFPI-2) expression by lysine-specific demethylase 1 and 2 (LSD1 and LSD2).
P2860

Synthesis and biological activity of optically active NCL-1, a lysine-specific demethylase 1 selective inhibitor.

Item
http://www.wikidata.org/entity/Q39608783
description
2010 nî lūn-bûn
@nan
2010年の論文
@ja
2010年論文
@yue
2010年論文
@zh-hant
2010年論文
@zh-hk
2010年論文
@zh-mo
2010年論文
@zh-tw
2010年论文
@wuu
2010年论文
@zh
2010年论文
@zh-cn
name
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@en
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@nl
type
label
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@en
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@nl
prefLabel
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@en
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@nl
P1433
P1476
P2093
P304
P31
P356
P407
P433
P478
P577
P698
P356
P1433
P1476
Synthesis and biological activ ...... thylase 1 selective inhibitor.
@en
P2093
P304
P31
P356
P407
P433
P478
P577
P698