Synthesis, structure-activity relationship, and pharmacophore modeling studies of pyrazole-3-carbohydrazone derivatives as dipeptidyl peptidase IV inhibitors.

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Optimization of pyrazole-containing 1,2,4-triazolo-[3,4-b]thiadiazines, a new class of STAT3 pathway inhibitors Antimicrobial screening and one-pot synthesis of 4-(substituted-anilinomethyl)-3-(2-naphthyl)-1-phenyl-1H-pyrazole derivatives

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P2860

Synthesis, structure-activity relationship, and pharmacophore modeling studies of pyrazole-3-carbohydrazone derivatives as dipeptidyl peptidase IV inhibitors.

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http://www.wikidata.org/entity/Q39646093

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2012 nî lūn-bûn

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2012年の論文

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2012年論文

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2012年論文

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2012年論文

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2012年論文

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2012年論文

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2012年论文

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2012年论文

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2012年论文

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name

Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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Synthesis, structure-activity ...... tidyl peptidase IV inhibitors.

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P1476

Synthesis, structure-activity ...... ptidyl peptidase IV inhibitors

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P2093

Cui Li

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Deyan Wu

http://www.w3.org/2001/XMLSchema#string

Fangfang Jin

http://www.w3.org/2001/XMLSchema#string

Guixia Liu

http://www.w3.org/2001/XMLSchema#string

Hualiang Jiang

http://www.w3.org/2001/XMLSchema#string

Jian Li

http://www.w3.org/2001/XMLSchema#string

Jin Zhu

http://www.w3.org/2001/XMLSchema#string

Wei Wang

http://www.w3.org/2001/XMLSchema#string

Yun Tang

http://www.w3.org/2001/XMLSchema#string

P2860

Rational design of a novel, potent, and orally bioavailable cyclohexylamine DPP-4 inhibitor by application of molecular modeling and X-ray crystallography of sitagliptin

Discovery of alogliptin: a potent, selective, bioavailable, and efficacious inhibitor of dipeptidyl peptidase IV

8-(3-(R)-aminopiperidin-1-yl)-7-but-2-ynyl-3-methyl-1-(4-methyl-quinazolin-2-ylmethyl)-3,7-dihydropurine-2,6-dione (BI 1356), a highly potent, selective, long-acting, and orally bioavailable DPP-4 inhibitor for the treatment of type 2 diabetes

Dipeptidyl-peptidase IV hydrolyses gastric inhibitory polypeptide, glucagon-like peptide-1(7-36)amide, peptide histidine methionine and is responsible for their degradation in human serum

Discovery and preclinical profile of Saxagliptin (BMS-477118): a highly potent, long-acting, orally active dipeptidyl peptidase IV inhibitor for the treatment of type 2 diabetes

Type 2 diabetes--therapy with dipeptidyl peptidase IV inhibitors.

CD26: a multifunctional integral membrane and secreted protein of activated lymphocytes.

A three-dimensional pharmacophore model for dipeptidyl peptidase IV inhibitors.

1-[[(3-hydroxy-1-adamantyl)amino]acetyl]-2-cyano-(S)-pyrrolidine: a potent, selective, and orally bioavailable dipeptidyl peptidase IV inhibitor with antihyperglycemic properties.

Pyrazole derivatives as partial agonists for the nicotinic acid receptor.

P304

897-906

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scholarly article

P356

10.1111/J.1747-0285.2012.01365.X

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P433

http://www.w3.org/2001/XMLSchema#string

P478

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Weiqiang Lu

Jin Huang

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2012-03-21T00:00:00Z

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P698

22381062

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Synthesis, structure-activity relationship, and pharmacophore modeling studies of pyrazole-3-carbohydrazone derivatives as dipeptidyl peptidase IV inhibitors.

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P2860

P2860

Synthesis, structure-activity relationship, and pharmacophore modeling studies of pyrazole-3-carbohydrazone derivatives as dipeptidyl peptidase IV inhibitors.

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