Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors.

Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors.

Item
http://www.wikidata.org/entity/Q40764005
The endocannabinoid system as an emerging target of pharmacotherapyEvidence against the presence of an anandamide transporterAnandamide transport is independent of fatty-acid amide hydrolase activity and is blocked by the hydrolysis-resistant inhibitor AM1172.Inhibition of monoacylglycerol lipase and fatty acid amide hydrolase by analogues of 2-arachidonoylglycerolThe endocannabinoid system: a general view and latest additionsThe endocannabinoid system: physiology and pharmacology.Studies of anandamide accumulation inhibitors in cerebellar granule neurons: comparison to inhibition of fatty acid amide hydrolaseThe cannabinoid system and its pharmacological manipulation--a review, with emphasis upon the uptake and hydrolysis of anandamide.Role of the cannabinoid system in pain control and therapeutic implications for the management of acute and chronic pain episodes.Endocannabinoid metabolism and uptake: novel targets for neuropathic and inflammatory pain.A systems pharmacology perspective on the clinical development of Fatty Acid amide hydrolase inhibitors for pain.Characterization of an anandamide degradation system in prostate epithelial PC-3 cells: synthesis of new transporter inhibitors as tools for this study.Actions of the endocannabinoid transport inhibitor AM404 in neuropathic and inflammatory pain models.The Endocannabinoid Reuptake Inhibitor WOBE437 Is Orally Bioavailable and Exerts Indirect Polypharmacological Effects via Different Endocannabinoid Receptors.
P2860

Design, synthesis and biological evaluation of novel arachidonic acid derivatives as highly potent and selective endocannabinoid transporter inhibitors.

Item
http://www.wikidata.org/entity/Q40764005
description
2001 nî lūn-bûn
@nan
2001年の論文
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2001年学术文章
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2001年学术文章
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2001年学术文章
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2001年学术文章
@zh-my
2001年学术文章
@zh-sg
2001年學術文章
@yue
2001年學術文章
@zh
2001年學術文章
@zh-hant
name
Design, synthesis and biologic ...... binoid transporter inhibitors.
@en
type
label
Design, synthesis and biologic ...... binoid transporter inhibitors.
@en
prefLabel
Design, synthesis and biologic ...... binoid transporter inhibitors.
@en
P1433
P1476
P2093
P304
P31
P356
P407
P433
P478
P50
P577
P698
P921
P356
P1433
P1476
Design, synthesis and biologic ...... abinoid transporter inhibitors
@en
P2093
P304
P31
P356
P407
P433
P478
P50
P577
P698
P921