Activation and block of recombinant GABA(A) receptors by pentobarbitone: a single-channel study.
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Structural studies of the actions of anesthetic drugs on the γ-aminobutyric acid type A receptorPregnenolone sulfate block of GABA(A) receptors: mechanism and involvement of a residue in the M2 region of the alpha subunitModulation of GABA(A) receptor channel gating by pentobarbitalCorrection for Inhibition Leads to an Allosteric Co-Agonist Model for Pentobarbital Modulation and Activation of α1β3γ2L GABAA ReceptorsPoint mutation in the first transmembrane region of the beta 2 subunit of the gamma--aminobutyric acid type A receptor alters desensitization kinetics of gamma--aminobutyric acid- and anesthetic-induced channel gatingThe dual modulatory effects of efavirenz on GABAA receptors are mediated via two distinct sites.Olfactory Hallucinations without Clinical Motor Activity: A Comparison of Unirhinal with Birhinal PhantosmiaPharmacological and anatomical evidence for an interaction between mGluR5- and GABA(A) alpha1-containing receptors in the discriminative stimulus effects of ethanol.m-Azipropofol (AziPm) a photoactive analogue of the intravenous general anesthetic propofolHow theories evolved concerning the mechanism of action of barbiturates.Anesthetic sites and allosteric mechanisms of action on Cys-loop ligand-gated ion channels.Structural link between γ-aminobutyric acid type A (GABAA) receptor agonist binding site and inner β-sheet governs channel activation and allosteric drug modulationAgonist-specific conformational changes in the α1-γ2 subunit interface of the GABA A receptor.A conserved salt bridge critical for GABA(A) receptor function and loop C dynamics.Distinct structural changes in the GABAA receptor elicited by pentobarbital and GABA.Molecular basis for modulation of recombinant alpha1beta2gamma2 GABAA receptors by protons.Activation of GABA(A) receptors containing the alpha4 subunit by GABA and pentobarbital.A novel mechanism of modulation of 5-HT₃A receptors by hydrocortisone.Pentobarbital produces activation and block of {alpha}1{beta}2{gamma}2S GABAA receptors in rapidly perfused whole cells and membrane patches: divergent results can be explained by pharmacokineticsMolecular basis of the differential sensitivity of nematode and mammalian muscle to the anthelmintic agent levamisole.The general anesthetic pentobarbital slows desensitization and deactivation of the glycine receptor in the rat spinal dorsal horn neurons.The GABAA receptor alpha 1 subunit Pro174-Asp191 segment is involved in GABA binding and channel gating.Benzodiazepines block alpha2-containing inhibitory glycine receptors in embryonic mouse hippocampal neurons.Conductance of GABAA channels activated by pentobarbitone in hippocampal neurons from newborn rats.Conformational changes at benzodiazepine binding sites of GABA(A) receptors detected with a novel technique.Contrasting actions of a convulsant barbiturate and its anticonvulsant enantiomer on the α1 β3 γ2L GABAA receptor account for their in vivo effects.A neurosteroid potentiation site can be moved among GABAA receptor subunits.Allosteric Modulation of αβδ GABAA Receptors.
P2860
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P2860
Activation and block of recombinant GABA(A) receptors by pentobarbitone: a single-channel study.
description
2000 nî lūn-bûn
@nan
2000年の論文
@ja
2000年論文
@yue
2000年論文
@zh-hant
2000年論文
@zh-hk
2000年論文
@zh-mo
2000年論文
@zh-tw
2000年论文
@wuu
2000年论文
@zh
2000年论文
@zh-cn
name
Activation and block of recombinant GABA
@nl
Activation and block of recomb ...... itone: a single-channel study.
@en
type
label
Activation and block of recombinant GABA
@nl
Activation and block of recomb ...... itone: a single-channel study.
@en
prefLabel
Activation and block of recombinant GABA
@nl
Activation and block of recomb ...... itone: a single-channel study.
@en
P2860
P356
P1476
Activation and block of recomb ...... itone: a single-channel study.
@en
P2093
P2860
P304
P356
10.1038/SJ.BJP.0703335
P407
P577
2000-05-01T00:00:00Z