Determination of the amino acid residue involved in [3H]beta-funaltrexamine covalent binding in the cloned rat mu-opioid receptor.
about
The evolution of vertebrate opioid receptorsCrystal structure of the µ-opioid receptor bound to a morphinan antagonistThe role of the hydrophilic Asn230 residue of the mu-opioid receptor in the potency of various opioid agonistsBrain region-specific N-glycosylation and lipid rafts association of the rat mu opioid receptorMutational analysis of the structure and function of opioid receptors.Opioid receptor three-dimensional structures from distance geometry calculations with hydrogen bonding constraints.Homology modeling of opioid receptor-ligand complexes using experimental constraintsGlial-restricted precursors: patterns of expression of opioid receptors and relationship to human immunodeficiency virus-1 Tat and morphine susceptibility in vitro.K303⁶·⁵⁸ in the μ opioid (MOP) receptor is important in conferring selectivity for covalent binding of β-funaltrexamine (β-FNA).Co-expression of GRK2 reveals a novel conformational state of the µ-opioid receptorThe opioid antagonist, β-funaltrexamine, inhibits NF-κB signaling and chemokine expression in human astrocytes and in miceMolecular recognition of opioid receptor ligands.Conformationally constrained opioid ligands: the Dmt-Aba and Dmt-Aia versus Dmt-Tic scaffoldDual labeled peptides as tools to study receptors: nanomolar affinity derivatives of TIPP (Tyr-Tic-Phe-Phe) containing an affinity label and biotin as probes of delta opioid receptors.Grand opening of structure-guided design for novel opioids.Consensus 3D model of μ-opioid receptor ligand efficacy based on a quantitative Conformationally Sampled Pharmacophore.A pharmacological comparison of the cloned frog and human mu opioid receptors reveals differences in opioid affinity and function.Fumaroylamino-4,5-epoxymorphinans and related opioids with irreversible μ opioid receptor antagonist effectsDiscovery of dermorphin-based affinity labels with subnanomolar affinity for mu opioid receptors.mu-opioid receptors are present in vagal afferents and their dendritic targets in the medial nucleus tractus solitarius.beta-Funaltrexamine, a gauge for the recognition site of wildtype and mutant H297Q mu-opioid receptors.An affinity label for delta-opioid receptors derived from [D-Ala2]deltorphin I.Characterization of functional μ opioid receptor turnover in rat locus coeruleus: an electrophysiological and immunocytochemical study.Molecular modeling study of the opioid receptor interactions with series of cyclic deltorphin analogues.Palmitoylation of the rat mu opioid receptor.
P2860
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P2860
Determination of the amino acid residue involved in [3H]beta-funaltrexamine covalent binding in the cloned rat mu-opioid receptor.
description
1996 nî lūn-bûn
@nan
1996年の論文
@ja
1996年学术文章
@wuu
1996年学术文章
@zh-cn
1996年学术文章
@zh-hans
1996年学术文章
@zh-my
1996年学术文章
@zh-sg
1996年學術文章
@yue
1996年學術文章
@zh
1996年學術文章
@zh-hant
name
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@en
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@nl
type
label
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@en
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@nl
prefLabel
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@en
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@nl
P2093
P2860
P356
P1476
Determination of the amino aci ...... cloned rat mu-opioid receptor.
@en
P2093
DesJarlais RL
Liu-Chen LY
Raveglia LF
P2860
P304
21422-21429
P356
10.1074/JBC.271.35.21422
P407
P577
1996-08-01T00:00:00Z