Uptake inhibitors but not substrates induce protease resistance in extracellular loop two of the dopamine transporter.
about
Hypoinsulinemia regulates amphetamine-induced reverse transport of dopamineRecognition of psychostimulants, antidepressants, and other inhibitors of synaptic neurotransmitter uptake by the plasma membrane monoamine transportersLow and high cocaine locomotor responding male Sprague-Dawley rats differ in rapid cocaine-induced regulation of striatal dopamine transporter function.Impaired striatal Akt signaling disrupts dopamine homeostasis and increases feeding.Syntaxin 1A regulates dopamine transporter activity, phosphorylation and surface expression.Palmitoylation controls dopamine transporter kinetics, degradation, and protein kinase C-dependent regulationMutational analysis of the high-affinity zinc binding site validates a refined human dopamine transporter homology modelAntagonist-induced conformational changes in dopamine transporter extracellular loop two involve residues in a potential salt bridgeDopamine transporter phosphorylation site threonine 53 regulates substrate reuptake and amphetamine-stimulated efflux.Reciprocal Phosphorylation and Palmitoylation Control Dopamine Transporter Kinetics.Phosphorylation of dopamine transporter serine 7 modulates cocaine analog binding.Comparative modeling of the human monoamine transporters: similarities in substrate binding.Tyr-95 and Ile-172 in transmembrane segments 1 and 3 of human serotonin transporters interact to establish high affinity recognition of antidepressants.Akt-dependent and isoform-specific regulation of dopamine transporter cell surface expression.Psychoactive substrates stimulate dopamine transporter phosphorylation and down-regulation by cocaine-sensitive and protein kinase C-dependent mechanisms.Phorbol ester induced trafficking-independent regulation and enhanced phosphorylation of the dopamine transporter associated with membrane rafts and cholesterol.Dopamine transporter phosphorylation site threonine 53 is stimulated by amphetamines and regulates dopamine transport, efflux, and cocaine analog binding.Localization of cocaine analog [125I]RTI 82 irreversible binding to transmembrane domain 6 of the dopamine transporter.
P2860
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P2860
Uptake inhibitors but not substrates induce protease resistance in extracellular loop two of the dopamine transporter.
description
2004 nî lūn-bûn
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2004年の論文
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2004年学术文章
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2004年学术文章
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2004年学术文章
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2004年学术文章
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2004年学术文章
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2004年學術文章
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2004年學術文章
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name
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@en
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@nl
type
label
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@en
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@nl
prefLabel
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@en
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@nl
P356
P1476
Uptake inhibitors but not subs ...... o of the dopamine transporter.
@en
P2093
Jon D Gaffaney
Roxanne A Vaughan
P304
P356
10.1124/MOL.65.3.692
P577
2004-03-01T00:00:00Z