Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics.
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18F-Labeled Single-Stranded DNA Aptamer for PET Imaging of Protein Tyrosine Kinase-7 ExpressionPET neuroimaging studies of [(18)F]CABS13 in a double transgenic mouse model of Alzheimer's disease and nonhuman primatesRadiochemistry on electrodes: Synthesis of an 18F-labelled and in vivo stable COX-2 inhibitor.Synthesis and preliminary PET imaging of 11C and 18F isotopologues of the ROS1/ALK inhibitor lorlatinibDifluorocarbene-Derived Trifluoromethylthiolation and [(18)F]Trifluoromethylthiolation of Aliphatic ElectrophilesOrtho-Stabilized (18) F-Azido Click Agents and their Application in PET Imaging with Single-Stranded DNA Aptamers.Efficient automated syntheses of high specific activity 6-[18F]fluorodopamine using a diaryliodonium salt precursorPreparation of o-Fluorophenols from Nonaromatic Precursors: Mechanistic Considerations for Adaptation to Fluorine-18 Radiolabeling.A Transmetalation Reaction Enables the Synthesis of [18F]5-Fluorouracil from [18F]Fluoride for Human PET ImagingIodonium ylide-mediated radiofluorination of 18F-FPEB and validation for human use[(18)F]6-fluoro-3,4-dihydroxy-L-phenylalanine--recent modern syntheses for an elusive radiotracer.Considerations in the Development of Reversibly Binding PET Radioligands for Brain Imaging.Fluorine-18 patents (2009-2015). Part 2: new radiochemistry.Fluorine-18 labelled building blocks for PET tracer synthesis.Sulfonium salts as leaving groups for aromatic labelling of drug-like small molecules with fluorine-18.Synthesis of (18) F-Difluoromethylarenes from Aryl (Pseudo) HalidesCu-Mediated C-H 18F-Fluorination of Electron-Rich (Hetero)arenesMild silver-mediated geminal difluorination of styrenes using an air- and moisture-stable fluoroiodane reagent.A Facile Radiolabeling of [18F]FDPA via Spirocyclic Iodonium Ylides: Preliminary PET Imaging Studies in Preclinical Models of NeuroinflammationCopper-Mediated Radiofluorination of Arylstannanes with [18F]KF.An automated synthesizer for electrochemical 18F-fluorination of organic compounds.Radiosynthesis and preliminary PET evaluation of (18)F-labeled 2-(1-(3-fluorophenyl)-2-oxo-5-(pyrimidin-2-yl)-1,2-dihydropyridin-3-yl)benzonitrile for imaging AMPA receptors.Efficient Pathway for the Preparation of Aryl(isoquinoline)iodonium(III) Salts and Synthesis of Radiofluorinated Isoquinolines.Mechanistic Studies and Radiofluorination of Structurally Diverse Pharmaceuticals with Spirocyclic Iodonium(III) Ylides.18F-Deoxyfluorination of Phenols via Ru π-ComplexesMolecular Imaging of Hydrolytic Enzymes Using PET and SPECT.Synthesis of (18)F-Arenes from Spirocyclic Iodonium(III) Ylides via Continuous-Flow MicrofluidicsSynthesis of meta-substituted [(18)F]3-fluoro-4-aminopyridine via direct radiofluorination of pyridine N-oxides.Late-stage [(18)F]Fluorination: New Solutions to Old ProblemsSynthesis of [18F]Arenes via the Copper-Mediated [18F]Fluorination of Boronic Acids.Novel 18F-Labeled κ-Opioid Receptor Antagonist as PET Radiotracer: Synthesis and In Vivo Evaluation of 18F-LY2459989 in Nonhuman Primates.Synthesis of [18 F]Fluoroarenes by Nucleophilic Radiofluorination of N-Arylsydnones.C(sp³)-¹⁸F bond formation by transition-metal-based [¹⁸F]fluorination.Brain Penetration of the ROS1/ALK Inhibitor Lorlatinib Confirmed by PET.Organocatalyst-assisted Ar-18F bond formation: a universal procedure for direct aromatic radiofluorination.Iodine-doped sumanene and its application for the synthesis of chalcogenasumanenes and silasumanenes.[18F]Fluorophenylazocarboxylates: Design and Synthesis of Potential Radioligands for Dopamine D3 and μ-Opioid Receptor.Synthesis of a Potent Aminopyridine-Based nNOS-Inhibitor by Two Recent No-Carrier-Added (18)F-Labelling Methods.18F-Labelling of electron rich iodonium ylides: application to the radiosynthesis of potential 5-HT2A receptor PET ligands.In Vitro and in Vivo Evaluation of 11C-Labeled Azetidinecarboxylates for Imaging Monoacylglycerol Lipase by PET Imaging Studies.
P2860
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P2860
Spirocyclic hypervalent iodine(III)-mediated radiofluorination of non-activated and hindered aromatics.
description
2014 nî lūn-bûn
@nan
2014年の論文
@ja
2014年学术文章
@wuu
2014年学术文章
@zh
2014年学术文章
@zh-cn
2014年学术文章
@zh-hans
2014年学术文章
@zh-my
2014年学术文章
@zh-sg
2014年學術文章
@yue
2014年學術文章
@zh-hant
name
Spirocyclic hypervalent iodine
@nl
Spirocyclic hypervalent iodine ...... ivated and hindered aromatics.
@en
type
label
Spirocyclic hypervalent iodine
@nl
Spirocyclic hypervalent iodine ...... ivated and hindered aromatics.
@en
prefLabel
Spirocyclic hypervalent iodine
@nl
Spirocyclic hypervalent iodine ...... ivated and hindered aromatics.
@en
P2093
P2860
P356
P1476
Spirocyclic hypervalent iodine ...... tivated and hindered aromatics
@en
P2093
Neil Vasdev
Nickeisha A Stephenson
Steven H Liang
P2860
P2888
P356
10.1038/NCOMMS5365
P407
P577
2014-07-09T00:00:00Z